Medicinal & Biomolecular Chemistry Concept

subject area of

• 1,4-Dihydropyridine Scaffold in Medicinal Chemistry, The Story So Far And Perspectives (Part 2): Action in Other Targets and Antitargets  Journal Articles
• 1,4-Dihydropyridine Scaffold in Medicinal Chemistry, The Story so Far And Perspectives (Part 1): Action in Ion Channels and GPCRs  Journal Articles
• 1-Triacontanol cerotate; isolated from Marsilea quadrifolia Linn. ameliorates reactive oxidative damage in the frontal cortex and hippocampus of chronic epileptic rats  Journal Articles
• 2-[F-18] FLUORO-L-DOPA  Conferences
• 2015 American college of rheumatology guideline for the treatment of rheumatoid arthritis.  Journal Articles
• 4-Aryl-3-(hydroxyalkyl)quinolin-2-ones:  Novel Maxi-K Channel Opening Relaxants of Corporal Smooth Muscle Targeted for Erectile Dysfunction  Journal Articles
• Pseudomonas Aeruginosa : Targeting Cell-Wall Metabolism for New Antibacterial Discovery and Development  Journal Articles
• A 2.13 Å Structure of E. coli Dihydrofolate Reductase Bound to a Novel Competitive Inhibitor Reveals a New Binding Surface Involving the M20 Loop Region  Journal Articles
• A Bone-Seeking trans-Cyclooctene for Pretargeting and Bioorthogonal Chemistry: A Proof of Concept Study Using ^99mTc- and ¹⁷⁷Lu-Labeled Tetrazines  Journal Articles
• A F-18 Labeling Strategy for Near Infrared Fluorophores. Multi-Modal Probes for Reactive Oxygen Species  Conferences
• A High-Throughput Screen of the GTPase Activity of Escherichia coli EngA to Find an Inhibitor of Bacterial Ribosome Biogenesis  Journal Articles
• A NEW STRATEGY FOR LABELING BIOMOLECULES THAT CONTAIN DISULFIDE BONDS WITH RHENIUM AND TECHNETIUM  Conferences
• A NEW STRATEGY FOR THE PREPARATION AND PURIFICATION OF TC-BASED RADIOPHARMACEUTICALS  Conferences
• A New Generation of M(I) Chelates for Correlating in vitro and in vivo Imaging  Conferences
• A New Series of Succinimido-ferrociphenols and Related Heterocyclic Species Induce Strong Antiproliferative Effects, Especially against Ovarian Cancer Cells Resistant to Cisplatin  Journal Articles
• A New Strategy To Improve the Metabolic Stability of Lactone: Discovery of (20S,21S)-21-Fluorocamptothecins as Novel, Hydrolytically Stable Topoisomerase I Inhibitors  Journal Articles
• A New Strategy for Labeling Unreactive Peptides and Proteins with N-Succinimidyl 4-[F-18]Fluorobenzoate ([F-18]SFB) using water-in-oil microemulsions  Conferences
• A Refined Model for the Somatostatin Pharmacophore:  Conformational Analysis of Lanthionine−Sandostatin Analogs  Journal Articles
• A Versatile Cell Death Screening Assay Using Dye-Stained Cells and Multivariate Image Analysis  Journal Articles
• A cell-based approach to characterize antimicrobial compounds through kinetic dose response  Journal Articles
• A comparative study of the in vivo behaviour of [¹⁸F] 2‐, 5‐ and 6‐fluoro‐L‐dopa in the human brain  Journal Articles
• A hybrid solid‐fluorous phase radioiodination and purification platform  Journal Articles
• A macrophage-stimulating compound from a screen of microbial natural products  Journal Articles
• A new system for profiling drug-induced calcium signal perturbation in human embryonic stem cell-derived cardiomyocytes.  Journal Articles
• A synthesis of 3-deoxydihydrolycoricidine: Refinement of a structurally minimum pancratistatin pharmacophore  Journal Articles
• A systematic review of the efficacy and safety of turmeric in the treatment of digestive disorders  Journal Articles
• A tribute to Leo C Vining  Journal Articles
• ACHIEVEING HIGH (APPARENT) SPECIFIC ACTIVITY FORMULATIONS USING FLUOROUS-PHASE CHEMISTRY  Conferences
• APPLICATION OF THE ONE‐DIMENSIONAL ISING MODEL TO THE SECONDARY STRUCTURES IN GLOBULAR PROTEINS.  Journal Articles
• AROMATIC RADIOFLUORINATION WITH [F-18] F2 IN ANHYDROUS HYDROGEN-FLUORIDE  Conferences
• Actions of two dopamine derivatives at adreno- and cholinoceptors  Journal Articles
• Alginate as an auxiliary bacterial membrane: binding of membrane-active peptides by polysaccharides  Journal Articles
• Alginate as an auxiliary bacterial membrane: binding of membrane‐active peptides by polysaccharides*  Journal Articles
• Allosteric Modulation of the Dopamine D₂ Receptor by Pro-Leu-Gly-NH₂ Peptidomimetics Constrained in Either a Polyproline II Helix or a Type II β-Turn Conformation  Journal Articles
• Allosteric Modulation of the Dopamine Receptor by Conformationally Constrained Type VI β-Turn Peptidomimetics of Pro-Leu-Gly-NH₂  Journal Articles
• Allosteric Sensing of Fatty Acid Binding by NMR: Application to Human Serum Albumin  Journal Articles
• An Endogenous Reactive Oxygen Species (ROS)‐Activated Histone Deacetylase Inhibitor Prodrug for Cancer Chemotherapy  Journal Articles
• Analog binding to melatonin receptors in chick brain: Effects of GTP and prazosin  Journal Articles
• Antagonists of the Calcium Receptor I. Amino Alcohol-Based Parathyroid Hormone Secretagogues  Journal Articles
• Anti-mesothelioma mechanism of action studies of a complex Cynara scolymus fraction using in silico target prediction and gene expression profiling  Conferences
• Antiallergic and antihistaminic effect of two extracts of Capparis spinosa L. flowering buds  Journal Articles
• Antibacterial Activity of Marine Bacterium Pseudomonas sp. Associated with Soft Coral Sinularia polydactyla against Streptococcus equi Subsp. zooepidemicus  Journal Articles
• Antibiotic and Antimalarial Quinones from Fungus-Growing Ant-Associated Pseudonocardia sp.  Journal Articles
• Antileishmanial macrolides from ant-associated Streptomyces sp. ISID311  Journal Articles
• Antimitotic activity of structurally simplified biaryl analogs of the anticancer agents colchicine and combretastatin A4  Journal Articles
• Antimitotic and cell growth inhibitory properties of combretastatin A-4-like ethers  Journal Articles
• Antineoplastic Agents. 362. Isolation and X-ray Crystal Structure of Dibromophakellstatin from the Indian Ocean Sponge Phakellia mauritiana  Journal Articles
• Antineoplastic Agents. 380. Isolation and X-ray Crystal Structure Determination of Isoaaptamine from the Republic of Singapore Hymeniacidon sp. and Conversion to the Phosphate Prodrug Hystatin 1  Journal Articles
• Antitussive, expectorant and anti-inflammatory activities of four alkaloids isolated from Bulbus of Fritillaria wabuensis.  Journal Articles
• Antitussive, expectorant and anti-inflammatory alkaloids from Bulbus Fritillariae Cirrhosae.  Journal Articles
• Apixaban  Journal Articles
• Apixaban (vol 33, pg 293, 2008)  Journal Articles
• Apocynum venetum leaf aqueous extract inhibits voltage-gated sodium channels of mouse neuroblastoma N2A cells  Journal Articles
• Apocynum venetum leaf extract, an antihypertensive herb, inhibits rat aortic contraction induced by angiotensin II: A nitric oxide and superoxide connection  Journal Articles
• Ascaridole-less infusions of Chenopodium ambrosioides contain a nematocide(s) that is(are) not toxic to mammalian smooth muscle  Journal Articles
• Assay and Drug Development Technologies  Journal
• Assessing the potential of using the Mo-100(p,2n)Tc-99m transformation as a means of producing Curie-quantities of Tc-99m on existing cyclotron infrastructure  Conferences
• BAY 43-9006: Early Clinical Data in Patients with Advanced Solid Malignancies  Journal Articles
• Bacillibactins E and F from a Marine Sponge-Associated Bacillus sp.  Journal Articles
• Bacillimidazoles A−F, Imidazolium-Containing Compounds Isolated from a Marine Bacillus  Journal Articles
• Bacterial proteases, untapped antimicrobial drug targets  Journal Articles
• Bacterial symbionts in agricultural systems provide a strategic source for antibiotic discovery  Journal Articles
• Bicyclic thiazolidine lactam peptidomimetics of the dopamine receptor modulating peptide Pro-Leu-Gly-NH2  Journal Articles
• Bioorganic and Medicinal Chemistry  Journal
• Bioorganic and Medicinal Chemistry Letters  Journal
• Biosynthesis of ebelactone A: isotopic tracer, advanced precursor and genetic studies reveal a thioesterase-independent cyclization to give a polyketide β-lactone  Journal Articles
• Biosynthesis of the piperidine alkaloids  Journal Articles
• Biotransformation of anticancer drugs by human and environmental microbiomes  Conferences
• Brevetoxin versus Brevenal Modulation of Human Nav1 Channels  Journal Articles
• CARBORANE DERIVATIVES FOR TARGETING Tc-99m TO NEURORECEPTORS  Conferences
• Characterization of the Isosteroidal Alkaloid Chuanbeinone from Bulbus of Fritillaria pallidiflora as Novel Antitumor Agent In Vitro and In Vivo.  Journal Articles
• ChemMedChem  Journal
• Chemical Biology and Drug Design  Journal
• Chemical variation from the neoantimycin depsipeptide assembly line  Journal Articles
• Chemistry and Biodiversity  Journal
• Chinese Traditional and Herbal Drugs  Journal
• Christopher Walsh: Pioneer and innovator in antibiotic and natural product chemical biology  Books
• Cite and oversight  Journal Articles
• Comparative pharmacological study of hydroethanol extracts of Passiflora alata and Passiflora edulis leaves†  Journal Articles
• Comparison of the interaction of methionine and norleucine‐containing peptides with phospholipid bilayers  Journal Articles
• Complementary and Alternative Medicine Use in Juvenile Idiopathic Arthritis: A Systematic Review of Prevalence and Evidence  Journal Articles
• Consideration of Cytokines as Therapeutics Agents or Targets  Journal Articles
• Correction to Preparation, Characterization, and Screening of a High Affinity Organometallic Probe for α-Adrenergic Receptors  Journal Articles
• Critical Role For Drug Delivery In The Development Of New Ophthalmic Treatments  Journal Articles
• Crocetin Prevents Dexamethasone-Induced Insulin Resistance in Rats  Journal Articles
• Crystal structure of tert.‐butyloxycarbonyl‐L‐prolyl‐D‐alanyl‐D‐alanyl‐N‐methylamide Dimeric β‐sheet formation  Journal Articles
• Current Drug Discovery Technologies  Journal
• Current Medicinal Chemistry  Journal
• Current Opinion in Drug Discovery and Development  Journal
• Current Pharmaceutical Design  Journal
• Current Signal Transduction Therapy  Journal
• Cytokine Therapeutics for Asthma: An Appraisal of Current Evidence and Future Prospects  Journal Articles
• Cytokines - Preface  Journal Articles
• Cytokines - Preface  Journal Articles
• Cytokines - Preface  Journal Articles
• Cytotoxic lanostane-type triterpenes from the fruiting bodies of Ganoderma lucidum.  Journal Articles
• DIRECT FLUORINATION OF MELATONIN AND 5-HYDROXY-L-TRYPTOPHAN WITH [F-18] F2  Conferences
• DISCOVERY AND EVALUATION OF A POTENTIAL MOLECULAR IMAGING AGENT FOR CATHEPSIN B  Conferences
• Deciphering the Diversified Metabolic Behavior of Hydroxyalkyl Ferrocidiphenols as Anticancer Complexes  Journal Articles
• Degradation of MAC13243 and studies of the interaction of resulting thiourea compounds with the lipoprotein targeting chaperone LolA  Journal Articles
• Design and Synthesis of Photoaffinity-Labeling Ligands of thel-Prolyl-l-leucylglycinamide Binding Site Involved in the Allosteric Modulation of the Dopamine Receptor  Journal Articles
• Design and synthesis of [ 125 I]Pyricoxib: A novel 125 I-labeled cyclooxygenase-2 (COX-2) inhibitors  Journal Articles
• Design, Synthesis, X-ray Analysis, and Dopamine Receptor-Modulating Activity of Mimics of the "C5" Hydrogen-Bonded Conformation in the Peptidomimetic 2-Oxo-3(R)-[(2(S)-pyrrolidinylcarbonyl)amino]-1-pyrrolidineacetamide  Journal Articles
• Design, Synthesis, and Dopamine Receptor Modulating Activity of Diketopiperazine Peptidomimetics ofl-Prolyl-l-leucylglycinamide  Journal Articles
• Design, Synthesis, and Dopamine Receptor Modulating Activity of Spiro Bicyclic Peptidomimetics ofl-Prolyl-l-leucyl-glycinamide  Journal Articles
• Design, synthesis and biological activity of piperlongumine derivatives as selective anticancer agents  Journal Articles
• Design, synthesis and biological evaluation of di-substituted noscapine analogs as potent and microtubule-targeted anticancer agents  Journal Articles
• Designing analogs of ticlopidine, a wall teichoic acid inhibitor, to avoid formation of its oxidative metabolites  Journal Articles
• Deterioration of storage phosphor screens with use  Journal Articles
• Determination of Productive Conformation of Acetylcholinesterase Substrates Using Molecular Mechanics  Journal Articles
• Determining the mode of action of bioactive compounds  Journal Articles
• Development and evaluation of a novel gallium-68 labelled pteroate for visualization of the folate receptor  Conferences
• Development of New Deoxycytidine Kinase Inhibitors and Noninvasive in Vivo Evaluation Using Positron Emission Tomography  Journal Articles
• Development of tag-free photoprobes for studies aimed at identifying the target of novel Group A Streptococcus antivirulence agents  Journal Articles
• Developments in mitogen-induced extracellular kinase 1 inhibitors and their use in the treatment of disease  Journal Articles
• Direct Factor Xa and direct thrombin inhibitors: a clinical trial update.  Journal Articles
• Direct fluorination of melatonin and 5-hydroxy-L-tryptophan with [18F]F2  Journal Articles
• Discovery of 1-arylpyrrolidone derivatives as potent p53–MDM2 inhibitors based on molecule fusing strategy  Journal Articles
• Discovery of HDAC6-Selective Inhibitor NN-390 with in Vitro Efficacy in Group 3 Medulloblastoma  Journal Articles
• Discovery of V-0219: A Small-Molecule Positive Allosteric Modulator of the Glucagon-Like Peptide-1 Receptor toward Oral Treatment for "Diabesity".  Journal Articles
• Discovery of a new class of cinnamyl-triazole as potent and selective inhibitors of aromatase (cytochrome P450 19A1)  Journal Articles
• Discovery of a novel class of aldol-derived 1,2,3-triazoles: Potent and selective inhibitors of human cytochrome P450 19A1 (aromatase)  Journal Articles
• Discovery of potent antiviral (HSV-1) quinazolinones and initial structure-activity relationship studies  Journal Articles
• Discovery of the Apoptosis-Inducing Activity and High Accumulation of the Butenolides, Menisdaurilide and Aquilegiolide, in Dicentra spectabilis  Journal Articles
• Diversity-oriented synthesis and bioactivity evaluation of N-substituted ferrocifen compounds as novel antiproliferative agents against TNBC cancer cells  Journal Articles
• Do Insecticides have Adverse Effects on Reproduction  Journal Articles
• Do the metabolites of 6-[F-18]fluoro-L-dopa and of [F-18]fluoro-meta-L-tyrosine contribute to the F-18 accumulation in the human brain?  Conferences
• Docking flexible ligands in proteins with a solvent exposure- and distance-dependent dielectric function  Journal Articles
• Dopamine receptor modulation by Pro-Leu-Gly-NH2 analogs possessing cyclic amino acid residues at the C-terminal position  Journal Articles
• Dopamine receptor modulation by a highly rigid spiro bicyclic peptidomimetic of Pro-Leu-Gly-NH2  Journal Articles
• Dopamine receptor modulation by conformationally constrained analogs of Pro-Leu-Gly-NH2  Journal Articles
• Drug Design and Discovery  Journal
• Drug Discovery Today  Journal
• Drug evaluation: AP-23573--an mTOR inhibitor for the treatment of cancer.  Journal Articles
• Drug evaluation: E-5564.  Journal Articles
• Drugs of the Future  Journal
• Dual-action peptides: a new strategy in the treatment of diabetes-associated neuropathy  Journal Articles
• Effect of Crude Methanol Extract ofTerminalia avicennioidesin Normal Gastric/Histamine-Induced HCl Secretions in Rats  Journal Articles
• Effect of a tobacco-related nitrosamine on intercellular communication in human urothelial cells: a possible factor in smoking-related bladder carcinogenesis.  Journal Articles
• Efficient Synthesis of Cannabigerol, Grifolin, and Piperogalin via Alumina-Promoted Allylation  Journal Articles
• Elcetrochemical nucleophilic radiofluorination of aromatic molecules  Conferences
• Electrowetting on dielectric digital microfluidic chips for multistep radiosynthesis of PET tracers  Conferences
• Emulsion reactors; A new platform for the synthesis of metal-based molecularimaging agents  Conferences
• Encapsulation of Radiolabeled Tetrazines in Pluronic F127 Nanoparticles for Pre-targeted SPECT Imaging and Radiotherapy using Bioorthogonal Chemistry  Conferences
• Endophthalmitis Prophylaxis in Cataract Surgery: Overview of Current Practice Patterns Around the World  Journal Articles
• Enzymatic synthesis of (−)-6-[18F]-fluoronorepinephrine from 6-[18F]-fluorodopamine by dopamine β-hydroxylase  Journal Articles
• Erratum to “Degradation of MAC13243 and studies of the interaction of resulting thiourea compounds with the lipoprotein targeting chaperone LolA” [Bioorg. Med. Chem. Lett. 23 (2013) 2426–2431]  Journal Articles
• European Journal of Medicinal Chemistry  Journal
• Evaluation of synthetic coumarins for antiausterity cytotoxicity against pancreatic cancers  Journal Articles
• Evidence-based support for phenotypic drug discovery in acute myeloid leukemia  Journal Articles
• Examining the correlations between GSK-3 inhibitory properties and anti-convulsant efficacy of valproate and valproate-related compounds  Journal Articles
• Excitation-contraction coupling mechanisms in airway smooth muscle: new targets in drug design.  Journal Articles
• Experimental Screening of Dihydrofolate Reductase Yields a “Test Set” of 50,000 Small Molecules for a Computational Data-Mining and Docking Competition  Journal Articles
• Expert Opinion on Therapeutic Patents  Journal
• Exploring the awareness of research among registered massage therapists in Ontario  Journal Articles
• Extracellular Signal-Regulated Kinases Modulate DNA Damage Response - A Contributing Factor to Using MEK Inhibitors in Cancer Therapy  Journal Articles
• Extremely Potent Block of Bacterial Voltage-Gated Sodium Channels by µ-Conotoxin PIIIA  Journal Articles
• F-18 LABELED XENON DIFLUORIDE  Conferences
• FLUORINE-18 LABELLED AROMATIC AMINO ACIDS FOR TUMOR IMAGING USING PET  Conferences
• Factors Promoting Tamoxifen Resistance in Breast Cancer via Stimulating Breast Cancer Stem Cell Expansion  Journal Articles
• First JA Medal goes to a paper on decalpenic acid  Journal Articles
• Fitoterapia  Journal
• Functional annotation of putative aminoglycoside antibiotic modifying proteins in Mycobacterium tuberculosis H37Rv  Journal Articles
• Future Medicinal Chemistry  Journal
• Garlic for hypertension: A systematic review and meta-analysis of randomized controlled trials  Journal Articles
• Gene Therapy, A Targeted Treatment for Diabetic Nephropathy  Journal Articles
• Gene Vectors for Cytokine Expression In Vivo  Journal Articles
• Gene set enrichment analysis and ingenuity pathway analysis to identify biomarkers in Sheng-ji Hua-yu formula treated diabetic ulcers  Journal Articles
• Ginkgo biloba extract for essential hypertension: A systemic review  Journal Articles
• Global Gastrointestinal Safety Profile of Etoricoxib and Lumiracoxib  Journal Articles
• Glycopeptide antibiotic biosynthesis  Journal Articles
• HUMAN TRANSFERRIN, ASIALOTRANSFERRIN AND THE INTERMEDIATE FORMS  Journal Articles
• High throughput screening identifies novel inhibitors of Escherichia coli dihydrofolate reductase that are competitive with dihydrofolate  Journal Articles
• Human Cytochrome P450 Liability Studies of trans-Dihydronarciclasine: A Readily Available, Potent, and Selective Cancer Cell Growth Inhibitor  Journal Articles
• Hydrophobic Interactions in Complexes of Antimicrobial Peptides with Bacterial Polysaccharides  Journal Articles
• IDrugs: the Investigational Drugs Journal  Journal
• INTERNATIONAL JOURNAL OF PHARMACOLOGY  Journal
• ISO-STRUCTURAL FLUORESCENT AND Tc-99m PROBES FOR LABELING BIOMOLECULES  Conferences
• Identification and Characterization of AES-135, a Hydroxamic Acid-Based HDAC Inhibitor That Prolongs Survival in an Orthotopic Mouse Model of Pancreatic Cancer  Journal Articles
• Identification of Small Molecule Chemical Inhibitors of the Collagen-Specific Chaperone Hsp47  Journal Articles
• Identification of amidoheteroaryls as potent inhibitors of mutant (V600E) B-Raf kinase with in vivo activity  Journal Articles
• Identification of common features within massage therapists’ professional identity  Journal Articles
• Identification of haemanthamine as a phytotoxic alkaloid in Narcissus pseudonarcissus L. (Daffodil) emerging buds  Journal Articles
• Ilodecakin. Schering-Plough Corp.  Journal Articles
• Imaging of Fibroblast Activation Protein in Cancer Xenografts Using Novel (4-Quinolinoyl)-glycyl-2-cyanopyrrolidine-Based Small Molecules  Journal Articles
• Imidazole-Fused Phenanthroline-Dyes for the Preparation of Multimodal Nuclear and Optical Imaging Probes  Conferences
• Immunology, Endocrine and Metabolic Agents in Medicinal Chemistry  Journal
• Impact of 5-HT3 receptor antagonists on peripheral and central diseases  Journal Articles
• Improved radiosynthesis and preliminary in vivo evaluation of the 11C-labeled tetrazine [11C]AE-1 for pretargeted PET imaging  Journal Articles
• In vitro biomass of Salvia corrugata: chemical analysis and evaluation of antimicrobial activity  Conferences
• In vitro evaluation of human cytochrome P450 and P-glycoprotein-mediated metabolism of some phytochemicals in extracts and formulations of African potato  Journal Articles
• Incorporation of an inducible nucleotide analog into DNA by DNA polymerases  Journal Articles
• Induction of GRP78 by valproic acid is dependent upon histone deacetylase inhibition  Journal Articles
• Induction of antimicrobial activities in heterologous streptomycetes using alleles of the Streptomyces coelicolor gene absA1  Journal Articles
• Informatic search for natural products (iSNAP) - A dereplication and discovery tool  Conferences
• Inhibition of the ANT(2″)-Ia resistance enzyme and rescue of aminoglycoside antibiotic activity by synthetic α-hydroxytropolones  Journal Articles
• Inhibitors of Bacterial Cystathionine β-Lyase:  Leads for New Antimicrobial Agents and Probes of Enzyme Structure and Function  Journal Articles
• Intedanib, a triple kinase inhibitor of VEGFR, FGFR and PDGFR for the treatment of cancer and idiopathic pulmonary fibrosis.  Journal Articles
• Integrated Network Pharmacology and Cellular Assay to Explore the Mechanisms of Selenized Tripterine Phytosomes (Se@Tri-PTs) Alleviating Podocyte Injury in Diabetic Nephropathy.  Journal Articles
• Integrating Complementary and Alternative Medicine With Primary Health Care Through Public Health To Improve Chronic Disease Management  Journal Articles
• Interaction of Calcium Channel Antagonists with Calcium: Structural Studies on Nicardipine and Its Ca2+ Complex  Journal Articles
• Interaction of calcium channel antagonists with calcium: spectroscopic and modeling studies on diltiazem and its Ca2+ complex  Journal Articles
• Interaction of calcium channel antagonists with calcium: structural studies on verapamil and its Ca2+ complex  Journal Articles
• Interaction of gonadotropin‐releasing hormone and its agonist analogs with Ca²⁺ in a nonpolar milieu. Correlation with biopotencies  Journal Articles
• Investigation of aryl halides as ketone bioisosteres: Refinement of potent and selective inhibitors of human cytochrome P450 19A1 (aromatase)  Journal Articles
• Invited Perspective: Screening in Academe: A Perspective on Implementation of University-Based Small Molecule Screening  Journal Articles
• Isolation and Synthesis of Veranamine, an Antidepressant Lead from the Marine Sponge Verongula rigida  Journal Articles
• Isolation of flavonoids from apple peel using novel graphene oxide cotton fiber  Journal Articles
• Isolation, Synthesis, and Semisynthesis of Amaryllidaceae Constituents from Narcissus and Galanthus sp.: De Novo Total Synthesis of 2-epi-Narciclasine  Journal Articles
• Isotopic labelling in mass spectrometry as a tool for studying reaction mechanisms of ion dissociations  Journal Articles
• Journal of Antibiotics  Journal
• Journal of Chemical Information and Modeling  Journal
• Journal of Complementary and Integrative Medicine  Journal
• Journal of Computer-Aided Molecular Design  Journal
• Journal of Ethnopharmacology  Journal
• Journal of Herbs, Spices and Medicinal Plants  Journal
• Journal of Labelled Compounds and Radiopharmaceuticals  Journal
• Journal of Medicinal Chemistry  Journal
• Journal of natural products  Journal
• L-prolyl-L-leucyl-glycinamide (PLG) and its analogs: Clinical implications in extrapyramidal motor disorders and depression  Journal Articles
• LCMS-based hierarchal clustering as a method to assess biosynthetic relationships among bacteria  Conferences
• Lanthionine−Somatostatin Analogs:  Synthesis, Characterization, Biological Activity, and Enzymatic Stability Studies  Journal Articles
• Lead Optimization of Positive Allosteric KV7.2/3 Channel Modulators toward Improved Balance of Lipophilicity and Aqueous Solubility.  Journal Articles
• Left Ventricular Non-compaction: From Recognition to Treatment  Journal Articles
• Ligands of Diltiazem Binding Site: An Overview of Some Chemotypes  Journal Articles
• Literature Search and Review  Journal Articles
• Machine Learning-Based Bioactivity Classification of Natural Products Using LC-MS/MS Metabolomics.  Journal Articles
• Macplocimine A, a new 18-membered macrolide isolated from the filamentous sulfur bacteria Thioploca sp.  Journal Articles
• Marine Drugs  Journal
• Material basis and mechanism of Descurainiae Semen Carbonisatum in treatment of acute lung injury based on nanotechnology  Journal Articles
• Mechanism of Action of an EPAC1-Selective Competitive Partial Agonist  Journal Articles
• Mechanisms of Specific versus Nonspecific Interactions of Aggregation-Prone Inhibitors and Attenuators  Journal Articles
• Medicinal Chemistry Research  Journal
• Medicinal Research Reviews  Journal
• Message from the Editors  Journal Articles
• Metabolomics, Metabonomics and Metabolite Profiling. Edited by William J. Griffiths.  Journal Articles
• Mini-Reviews in Medicinal Chemistry  Journal
• Modifier Gene Studies to Identify New Therapeutic Targets in Cystic Fibrosis  Journal Articles
• Modular pharmacology-based approach to identify hub genes and kernel pathways of taodan granules treated psoriasis  Journal Articles
• Modulation of Salmonella gene expression by subinhibitory concentrations of quinolones  Journal Articles
• Molecular Dynamics of Fibrinogen Adsorption onto Graphene, but Not onto Poly(ethylene glycol) Surface, Increases Exposure of Recognition Sites That Trigger Immune Response  Journal Articles
• Molecular Informatics  Journal
• Molecular Mechanism of Action and Selectivity of Sodium Ch annel Blocker Insecticides  Journal Articles
• N-demethylation of cyamemazine via non-classical Polonovski reaction and its conjugation to bovine serum albumin  Journal Articles
• Natural Product Research  Journal
• Natural products for the treatment of neurodegenerative diseases  Journal Articles
• Natural products in diabetes research: quantitative literature analysis.  Journal Articles
• New Anticoagulants for the Prevention of Thromboembolism  Journal Articles
• New phenolic inhibitors of yeast homoserine dehydrogenase  Journal Articles
• Oncology Research  Journal
• One Solution for All: Searching for Universal Aptamers for Constantly Mutating Spike Proteins of SARS‐CoV‐2  Journal Articles
• One-pot, multicomponent synthesis of 2,3-disubstituted quinazolin-ones with potent and selective activity against Toxoplasma gondii  Journal Articles
• Opinion: Direct-To-Consumer Advertising of Prescription Medicines: A Counter Argument  Journal Articles
• Ovarian Toxicity of Environmental Toxicants  Journal Articles
• PREPRINTS . AN OLD INFORMATION DEVICE WITH NEW OUTLOOKS  Conferences
• Panax quinquefolium saponin combined with dual antiplatelet drugs inhibits platelet adhesion to injured HUVECs via PI3K/AKT and COX pathways  Journal Articles
• Pancratistatin Selectively Induces Apoptosis in Cancer Cells and Reduces Growth of Colon Xenografts  Conferences
• Permutationally Invariant Deep Learning Approach to Molecular Fingerprinting with Application to Compound Mixtures  Journal Articles
• Pharmaceutical Biology  Journal
• Pharmacologic Properties of the New Oral Anticoagulants: A Clinician-oriented Review with a Focus on Perioperative Management  Journal Articles
• Pharmacological Treatment of Hypertension in Pregnancy  Journal Articles
• Pharmacology and Clinical Potential of Direct Thrombin Inhibitors  Journal Articles
• Phenylalkylamines in calcium channels: computational analysis of experimental structures  Journal Articles
• Phytomedicine  Journal
• Phytotherapy Research  Journal
• Planta Medica  Journal
• Polyphenolic natural products and natural product–inspired steroidal mimics as aromatase inhibitors  Journal Articles
• Portulaca oleracea extract reduces gut microbiota imbalance and inhibits colorectal cancer progression via inactivation of the Wnt/β-catenin signaling pathway  Journal Articles
• Potent and selective inhibition of human cytochrome P450 3A4 by seco-pancratistatin structural analogs  Journal Articles
• Potential Therapeutic Effects of Exogenous Ketone Supplementation for Type 2 Diabetes: A Review  Journal Articles
• Preparation and Evaluation of Carborane Analogues of Tamoxifen  Journal Articles
• Preparation and Evaluation of Fluorine-18-Labeled Insulin as a Molecular Imaging Probe for Studying Insulin Receptor Expression in Tumors  Journal Articles
• Preparation and Evaluation of Halogenated and Metallated Cathepsin B Inhibitors as Molecular Imaging Agents  Conferences
• Preparation and Evaluation of Radiolabeled Antibody Recruiting Small Molecules That Target Prostate-Specific Membrane Antigen for Combined Radiotherapy and Immunotherapy  Journal Articles
• Preparation and evaluation of reagents for tagging amino and thiol groups with fluorous stannanes. A convenient method for producing radioiodinated compounds in high effective specific activity  Journal Articles
• Preparation and in vivo testing of Tc-99m(I)-tetrazines for pretargeted imaging  Conferences
• Preparation of labelled 2‐methoxy‐3‐alkylpyrazines: synthesis and characterization of deuterated 2‐methoxy‐3‐isopropylyrazine and 2‐methoxy‐3‐isobutylpyrazine  Journal Articles
• Preparation of technetium‐99m bifunctional chelate complexes using a microfluidic reactor: a comparative study with conventional and microwave labeling methods  Journal Articles
• Preparation, Characterization, and Screening of a High Affinity Organometallic Probe for α-Adrenergic Receptors  Journal Articles
• Pretargeted PET Imaging of Bone Using a Trans-cyclooctene-Labeled Bisphosphonate  Conferences
• Proline‐containing β‐turns  Journal Articles
• Quantum Mechanics/Molecular Mechanics Strategies for Docking Pose Refinement: Distinguishing between Binders and Decoys in CytochromecPeroxidase  Journal Articles
• RADIOFLUORINATION OF L-THREO-3-(3,4-DIHYDROXYPHENYL)SERINE: SYNTHESIS OF POTENTIAL F-18 LABELLED PET TRACERS FOR NOREPINEPHRINE  Conferences
• RADIOFLUORINATION WITH XENON DIFLUORIDE - L-6[F-18]FLUORO-DOPA  Conferences
• REGIO- AND STEREOSELECTIVE ELECTROPHILIC FLUORINATION OF 3,4,6-TRI-O-ACETYL-D-GLUCAL (TAG) IN ACIDIC MEDIUM  Conferences
• Radiolabeled nanoscale gas vesicles using bioorthogonal chemistry for multimodal SPECT and ultrasound imaging  Conferences
• Radiosensitization of Colon Cancer Cell Lines by Docetaxel: Mechanisms of Action  Journal Articles
• Rank Ordering Plate Data Facilitates Data Visualization and Normalization in High-Throughput Screening  Journal Articles
• Re-evaluation of Fibrogenic Cytokines in Lung Fibrosis  Journal Articles
• Reactivity and radiochemical yield of [18F]F2 from 18O(p,n)18F target: 'SINGLE-SHOOT' vs 'DOUBLE-SHOOT' method for the production of [18F]F2  Conferences
• Repeated recovery, distillation and reuse of oxygen-18 water in 18O(p,n)18F high pressure target  Conferences
• Reproductive Toxicology of Environmental Toxicants: Emerging Issues and Concerns  Journal Articles
• Residual Vein Thrombosis and D-Dimer for Optimizing Duration of Anticoagulation in Idiopathic Deep Vein Thrombosis  Journal Articles
• Reversing Anticoagulant Therapy  Journal Articles
• Review of Cytotoxic CA4 Analogues that Do Not Target Microtubules: Implications for CA4 Development  Journal Articles
• Review of Cytotoxic CA4 Analogues that Do Not Target Microtubules: Implications for CA4 Development.  Journal Articles
• Role of DAP12 in Innate and Adaptive Immune Responses  Journal Articles
• Role of Dendritic Cell-Derived Cytokines in Immune Regulation  Journal Articles
• SLAS Discovery  Journal
• SYNTHESIS OF 18F-RADIOTRACERS IN HIGH SPECIFIC ACTIVITY USING THE FLUOROUS APPROACH  Conferences
• SYNTHESIS, ANTIFUNGAL AND ANTI-BACTERIAL ACTIVITY OF AMINOALKYL KETONES IN SULFUR HETEROCYCLIC SERIES  Journal Articles
• SYNTHESIS, RADIOLABELLING AND BIOLOGICAL EVALUATION OF TARGETED METALLACARBORANE (M=99MTc) DERIVATIVES FOR IMAGING NEURORECEPTORS  Conferences
• Safety and Efficacy of Ximelagatran: Meta-Analysis of the Controlled Randomized Trials for the Prophylaxis or Treatment of Venous Thromboembolism  Journal Articles
• Screening of ligands for redox-active europium using magnetic resonance imaging  Journal Articles
• Searching for Structure: Characterizing the Protein Conformational Landscape with Clustering-Based Algorithms.  Journal Articles
• Selective cytochrome P450 3A4 inhibitory activity of Amaryllidaceae alkaloids  Journal Articles
• Selectivity of [¹⁸F]F₂ towards L‐α‐methyltyrosine and L‐tyrosine: A radiochemical and NMR spectroscopic study  Journal Articles
• Sheng-ji Hua-yu ointment ameliorates cutaneous wound healing in diabetes via up-regulating CCN1  Journal Articles
• Side chain flexibility and the pore dimensions in the GABAA receptor  Journal Articles
• Silicon/Fluorine-18/PSMA: A winning team for PET imaging of prostate cancer  Conferences
• Simultaneous synthesis of 18F-labelled 6-fluoro-m-tyramine and 6-fluoro-3-hydroxy phenylacetic acid: 18F-containing metabolites of [18F]6-fluoro-m-tyrosine  Conferences
• Single amino acid chelate complexes of the M(CO)₃⁺ core for correlating fluorescence and radioimaging studies (M = ^99mTc or Re)  Journal Articles
• Small Structural Differences between Two Ferrocenyl Diphenols Determine Large Discrepancies of Reactivity and Biological Effects  Journal Articles
• Small molecule functional discrimination of the kinases required for the microbial synthesis of threonine and isoleucine  Journal Articles
• Small molecule immunomodulins from cultures of the human microbiome member Lactobacillus plantarum  Journal Articles
• Structural Insights into the Inhibition of Undecaprenyl Pyrophosphate Synthase from Gram-Positive Bacteria  Journal Articles
• Structural–Functional Studies of Burkholderia cenocepacia d-Glycero-β-d-manno-heptose 7-Phosphate Kinase (HldA) and Characterization of Inhibitors with Antibiotic Adjuvant and Antivirulence Properties  Journal Articles
• Structure-activity studies on N -Substituted tranylcypromine derivatives lead to selective inhibitors of lysine specific demethylase 1 (LSD1) and potent inducers of leukemic cell differentiation  Journal Articles
• Structure-activity-relationships of the Stability of Six Pentathiepins Towards Glutathione: Possible Correlations with Biological Activities.  Journal Articles
• Structures and biosynthesis of 12-membered macrocyclic depsipeptides from Streptomyces sp. ML55  Journal Articles
• Structure–activity studies on acetylcholinesterase inhibition in the lycorine series of Amaryllidaceae alkaloids  Journal Articles
• Structure–activity studies on seco-pancratistatin analogs: Potent inhibitors of human cytochrome P450 3A4  Journal Articles
• Studies directed towards the refinement of the pancratistatin cytotoxic pharmacophore  Journal Articles
• Synthesis and Biological Activity of a Focused Library of Mitogen‐activated Protein Kinase Phosphatase Inhibitors  Journal Articles
• Synthesis and Biological Evaluation of Fully Functionalized seco-Pancratistatin Analogues  Journal Articles
• Synthesis and Characterization of Rhenium and Technetium-99m Labeled Insulin  Journal Articles
• Synthesis and Dopamine Receptor Modulating Activity of 3-Substituted γ-Lactam Peptidomimetics of l-Prolyl-l-leucyl-glycinamide  Journal Articles
• Synthesis and Dopamine Receptor Modulating Activity of Novel Peptidomimetics ofl-Prolyl-l-leucyl-glycinamide Featuring α,α-Disubstituted Amino Acids  Journal Articles
• Synthesis and Dopamine Receptor Modulating Activity of Substituted Bicyclic Thiazolidine Lactam Peptidomimetics of l-Prolyl-l-leucyl-glycinamide  Journal Articles
• Synthesis and Evaluation of Anticancer Natural Product Analogues Based on Angelmarin: Targeting the Tolerance towards Nutrient Deprivation  Journal Articles
• Synthesis and Evaluation of Radioiodinated Acyloxymethyl Ketones as Activity-Based Probes for Cathepsin B  Journal Articles
• Synthesis and Preclinical Evaluation of [¹⁸F]SiFA-PSMA Inhibitors in a Prostate Cancer Model  Journal Articles
• Synthesis and Screening of Mono- and Di-Aryl Technetium and Rhenium Metallocarboranes. A New Class of Probes for the Estrogen Receptor  Journal Articles
• Synthesis and Structure–Activity Relationships of the First Ferrocenyl-Aryl-Hydantoin Derivatives of the Nonsteroidal Antiandrogen Nilutamide  Journal Articles
• Synthesis and Structure−Activity Relationships of Truncated Bisubstrate Inhibitors of Aminoglycoside 6‘-N-Acetyltransferases  Journal Articles
• Synthesis and biological characterisation of a series of iberiotoxin analogues  Journal Articles
• Synthesis and biological evaluation of analogs of Pro-Leu-Gly-NH2 modified at the leucyl residue  Journal Articles
• Synthesis and dopamine receptor modulating activity of lactam conformationally constrained analogs of Pro-Leu-Gly-NH2  Journal Articles
• Synthesis and dopamine receptor modulating activity of unsubstituted and substituted triproline analogues of l-prolyl-l-leucyl-glycinamide (PLG)  Journal Articles
• Synthesis and evaluation of photoaffinity probes directed at lanosterol 14α-demethylase (P-45014DM)  Journal Articles
• Synthesis and in Vitro Evaluation of¹⁸F- and¹⁹F-Labeled Insulin:  A New Radiotracer for PET-based Molecular Imaging Studies  Journal Articles
• Synthesis and inhibitory action on HMG-CoA synthase of racemic and optically active oxetan-2-ones (β-Lactones)  Journal Articles
• Synthesis and structure-activity relationships among glycosidic derivatives of 4'-demethylepipodophyllotoxin and epipodophyllotoxin, showing VM26- and VP16-213-like activities.  Journal Articles
• Synthesis of Pro-Leu-Gly-NH2 analogs modified at the prolyl residue and evaluation of their effects on the receptor binding activity of the central dopamine receptor agonist, ADTN  Journal Articles
• Synthesis of cholesteryl esters of labelled fatty acids  Journal Articles
• Synthesis of fluorine-18 labelled 5-fluoro-L-DOPA by direct fluorination of L-DOPA  Conferences
• Synthesis of f‐18 labelled fluoro‐melatonins and 5‐hydroxy‐fluoro‐tryptophans  Journal Articles
• Synthesis of non-nucleoside anti-viral cyclopropylcarboxacyl hydrazones and initial anti-HSV-1 structure-activity relationship studies  Journal Articles
• Synthesis of radiolabelled antibody recruiting small molecules (radio-ARMs) for combined radio and immune therapy using bioorthogonal chemistry  Conferences
• Synthesis of α-methylstilbenes using an aqueous Wittig methodology and application toward the development of potent human aromatase inhibitors  Journal Articles
• Synthetic Biology Facilitates Semisynthetic Development of Type V Glycopeptide Antibiotics Targeting Vancomycin-Resistant Enterococcus  Journal Articles
• Synthetic Glucocorticoids: Antenatal Administration and Long-term Implications  Journal Articles
• Systematic replacement of amides by 1,4-disubstituted[1,2,3]triazoles in Leu-enkephalin and the impact on the delta opioid receptor activity.  Journal Articles
• Systems Medicine Approaches for the Definition of Complex Phenotypes in Chronic Diseases and Ageing. From Concept to Implementation and Policies  Journal Articles
• TEMPERATURE EFFECT ON THE STEREOSPECIFICITY OF NUCLEOPHILIC FLUORINATION: FORMATION OF [18F]TRANS-4-FLUORO-L-PROLINE DURING THE SYNTHESIS OF [18F]CIS-4-FLUORO-L-PROLINE  Conferences
• THE MOLECULAR COMPONENTS OF HUMAN TRANSFERRIN TYPE C  Journal Articles
• THE PREPARATION AND IN VITRO EVALUATION OF CARBORANE SELECTIVE ESTROGEN RECEPTOR MODULATORS  Conferences
• Taking aim at wall teichoic acid synthesis: new biology and new leads for antibiotics  Journal Articles
• Targeting prostate-specific membrane antigen (PSMA) with F-18-labeled compounds: The influence of prosthetic groups on tumor uptake  Conferences
• Temperature effects on the stereospecificity of nucleophilic fluorination: formation of trans‐[¹⁸F]4‐fluoro‐l‐proline during the synthesis of cis‐[¹⁸F]4‐fluoro‐l‐proline  Journal Articles
• Tetrazine-Derived Near-Infrared Dye for Targeted Photoacoustic Imaging of Bone  Journal Articles
• The AMP-Activated Protein Kinase: Role in Regulation of Skeletal Muscle Metabolism and Insulin Sensitivity  Journal Articles
• The Effect of Prebiotic Products on Decreasing Adiposity Parameters in Overweight and Obese Individuals: A Systematic Review and Meta- Analysis  Journal Articles
• The Effects of Commercial Preparations of Herbal Supplements Commonly Used by Women on the Biotransformation of Fluorogenic Substrates by Human Cytochromes P450  Journal Articles
• The First Organometallic Selective Estrogen Receptor Modulators (SERMs) and Their Relevance to Breast Cancer  Journal Articles
• The Hunt for New Tuberculosis Vaccines: Anti-TB Immunity and Rational Design of Vaccines  Journal Articles
• The Identification of 5-Hydroxyl-L-norvaline in Cultures of Pyridoxine Auxotrophs of Escherichia coli B  Journal Articles
• The International Natural Product Sciences Taskforce (INPST) and the power of Twitter networking exemplified through #INPST hashtag analysis  Journal Articles
• The Role of IL-15 Signaling in the Induction of Innate Antiviral Responses  Journal Articles
• The discovery of rofecoxib, [MK 966, VIOXX®, 4-(4′-methylsulfonylphenyl)-3-phenyl-2(5H)-furanone], an orally active cyclooxygenase-2 inhibitor  Journal Articles
• The effectiveness and safety of Xiao'er Feike granules in the treatment of acute bronchitis: A systematic review and meta-analysis.  Journal Articles
• The effects of different concentrations of saffron (Crocus sativus) decoction on preterm delivery in mice  Conferences
• The inorganic crystal structure data base  Journal Articles
• The sequential production of [18F]-6-FDOPA and [18F]-F-m-tyrosine (or [18F]-2-FDG) from the same dilute [18F]F2 target gas  Conferences
• The total alkaloid fraction of bulbs of Fritillaria cirrhosa displays anti-inflammatory activity and attenuates acute lung injury.  Journal Articles
• Therapeutic Peptides: New Arsenal Against Drug Resistant Pathogens  Journal Articles
• Therapeutic advances in the treatment of osteoporosis  Journal Articles
• Therapeutic approaches for haemophilia  Journal Articles
• Therapeutic patents for the treatment of premenstrual syndrome and premenstrual dysphoric disorder: historical perspectives and future directions  Journal Articles
• Thermodynamic and NMR analysis of inhibitor binding to dihydrofolate reductase  Journal Articles
• Thiopeptides: antibiotics with unique chemical structures and diverse biological activities  Journal Articles
• Three new polyketides from fruiting bodies of the endophytic ascomyceteXylaria polymorpha  Journal Articles
• Tifacogin (Chiron Corp/Pharmacia Corp).  Journal Articles
• Triazole Appending Agent (TAAG): A new hydrophilic iodine-containing prosthetic group for the preparation of targeted radiopharmaceuticals  Conferences
• Trifluoromethanesulfonic acid, an alternative solvent medium for the direct electrophilic fluorination of DOPA: new syntheses of 6‐[¹⁸F]fluoro‐L‐DOPA and 6‐[¹⁸F]fluoro‐D‐DOPA  Journal Articles
• Tris(3-hydroxypropyl)phosphine (THPP): A mild, air-stable reagent for the rapid, reductive cleavage of small-molecule disulfides  Journal Articles
• Two New Nor‐seco‐Isodhilarane‐Type Meroterpenoids from the Endophytic Fungus Penicillium purpurogenum  Journal Articles
• Two approaches for the syntheis of carbon‐11 labeled (R) and (S)‐albuterol  Journal Articles
• Uptake of Fe III influences the topographical arrangement of N‐glycan(s) in human transferrin  Journal Articles
• Using chemical bonds to analyze data retrieved from the inorganic crystal structure database  Journal Articles
• Variation determinants within massage therapists’ professional identity  Journal Articles
• Winners of the 2013 JA Medals for excellence  Journal Articles
• Winners of the 2014 JA Medals for excellence  Journal Articles
• Zhongguo Zhongyao Zazhi  Journal
• [Exploration and practice of post-marketing survival benefit evaluation of Chinese patent medicine for cancer].  Journal Articles
• [F-18]Fluoro-meta-L-tyrosine is a better PET tracer than [F-18]fluoro-L-dopa for the deliniation of dopaminergic structures in the human brain  Conferences
• eta(5)-TYPE ORGANOMETALLIC COMPOUNDS AND THE PREPARATION OF Tc RADIOTRACERS  Conferences
• iso-Lactam and reduced amide analogues of the peptidomimetic dopamine receptor modulator 3(R)-[(2(S)-Pyrrolidinylcarbonyl)amino]-2-oxo-1-pyrrolidineacetamide  Journal Articles
• β-Lactone natural products and derivatives inactivate homoserine transacetylase, a target for antimicrobial agents  Journal Articles
• β‐STRUCTURE OF POLYPEPTIDES IN NON‐AQUEOUS SOLUTIONS: I. Spectral Characteristics of the Polypeptide Backbone  Journal Articles
• β‐STRUCTURE OF POLYPEPTIDES IN NON‐AQUEOUS SOLUTIONS: II. Side‐Chain Orientation  Journal Articles
• “I am a healthcare practitioner”: A qualitative exploration of massage therapists’ professional identity  Journal Articles
• “Just don’t be creepy”: A phenomenological study of the experiences of men in massage therapy  Journal Articles