Binding, Competitive Concept

subject area of

• 2-(Oxadiazolyl)- and 2-(thiazolyl)imidazo[1,2-a]pyrimidines as agonists and inverse agonists at benzodiazepine receptors  Academic Article
• 2-[125I]Iodomelatonin binding sites in the quail heart: Characteristics, distribution and modulation by guanine nucleotides and cations  Academic Article
• 2-[¹²⁵I]Iodomelatonin Binding in the Brains of Four Salmonids  Academic Article
• 3H-spiroperidol binding and dopamine-stimulated adenylate cyclase: Evidence for multiple classes of receptors in primate brain regions  Academic Article
• A Model for Agonism and Antagonism in an Ancient and Ubiquitous cAMP-binding Domain  Academic Article
• A PET study of effects of chronic 3,4-methylenedioxymethamphetamine (MDMA, “ecstasy”) on serotonin markers in Göttingen minipig brain  Academic Article
• A molecular defect in two families with hemolytic poikilocytic anemia: reduction of high affinity membrane binding sites for ankyrin.  Academic Article
• A simple and efficient method for solubilization of the dopamine receptor  Academic Article
• A simple and rapid competitive enzyme-linked immunosorbent assay to identify HPA-1a (PlA1)-negative donor platelet units  Academic Article
• A study of phosphoglycerate kinase in human erythrocytes  Academic Article
• Activation of a recombinant human factor VII structural analogue alters its affinity of binding to tissue factor  Academic Article
• Activation of protein C and thrombin activable fibrinolysis inhibitor on cultured human endothelial cells  Academic Article
• Active suppression of host-vs graft reaction in pregnant mice. IX. Soluble suppressor activity obtained from allopregnant mouse decidua that blocks the cytolytic effector response to IL-2 is related to transforming growth factor-beta.  Academic Article
• Active suppression of host-vs-graft reaction in pregnant mice. VI. Soluble suppressor activity obtained from decidua of allopregnant mice blocks the response to IL 2.  Academic Article
• Agonist binding fraction of dopamine D2/3 receptors in rat brain: A quantitative autoradiographic study  Academic Article
• Agonists Interaction with Radiolabeled α-Adrenoceptor Antagonists Binding Sites in Rat Mesenteric Artery  Academic Article
• Allosteric Modulation of the Dopamine D2Receptor by Pro-Leu-Gly-NH2Peptidomimetics Constrained in Either a Polyproline II Helix or a Type II β-Turn Conformation  Academic Article
• Alpha-2 adrenoceptors on nerves and muscles of rat uterus.  Academic Article
• Binding Sites for 2-[¹²⁵I]Iodomelatonin in the Adrenal Gland  Academic Article
• Binding of 125I-labelled human chorionic gonadotropin to cell membrane receptors in rabbit ovarian slices  Academic Article
• Biochemical studies on opioid and alpha 2-adrenergic receptors in canine submucosal neurons  Academic Article
• Calcium channel antagonist binding and pharmacology in rat uterine smooth muscle  Academic Article
• Calpain proteolysis of von Willebrand factor enhances its binding to platelet membrane glycoprotein IIb/IIIa: an explanation for platelet aggregation in thrombotic thrombocytopenic purpura  Academic Article
• Carbohydrate-binding Modules Recognize Fine Substructures of Cellulose  Academic Article
• Characteristics of [3H] propyl beta-carboline-3-carboxylate binding to benzodiazepine receptors in human brain.  Academic Article
• Characterization of High-Affinity Dopamine D2Receptors and Modulation of Affinity States by Guanine Nucleotides in Cholate-Solubilized Bovine Striatal Preparations  Academic Article
• Characterization of [3H]Ryanodine Binding Sites in Smooth Muscle of Dog Mesentery Artery  Academic Article
• Characterization of alpha 2 adrenoceptors and other adrenoceptors in membranes isolated from dog mesenteric nerve axons.  Academic Article
• Characterization of beta adrenoceptors on cultured endothelial cells by radioligand binding  Academic Article
• Characterization of cholecystokinin receptors in canine intestinal circular muscle  Academic Article
• Characterization of galanin receptor in canine small intestinal circular muscle synaptosomes  Academic Article
• Characterization of neurokinin type 1 receptor in canine small intestinal muscle  Academic Article
• Characterization of the prostanoid TP receptor population in human nonpregnant myometrium.  Academic Article
• Characterization of α-Adrenoceptors in Canine Mesenteric Vein  Academic Article
• Combination plots as graphical tools in the study of enzyme inhibition  Academic Article
• Comparative pharmacological properties and functional coupling of mu and delta opioid receptor sites in human neuroblastoma SH-SY5Y cells.  Academic Article
• Comparison of the Pharmacological Characteristics of 2-[¹²⁵I]Iodomelatonin Binding Sites in the Lung, Spleen, Brain and Kidney of Chicken  Academic Article
• Competitive Effects from an Artificial Tear Solution to Protein Adsorption  Academic Article
• Competitive solid-phase enzyme immunoassay for melatonin in human and rat serum and rat pineal gland.  Academic Article
• Complement receptor type three (CD11b/CD18) of human polymorphonuclear leukocytes recognizes fibrinogen.  Academic Article
• Complex formation of platelet thrombospondin with fibrinogen.  Academic Article
• Complex formation of platelet thrombospondin with histidine-rich glycoprotein.  Academic Article
• Confirmatory Testing Demonstrates That False-Positive Rates in the Chlamydiazyme Assay are Influenced by Gender and Genital Specimen Type  Academic Article
• Conformational determinants in receptor recognition of peptide hormones: interaction of parathyroid hormone with the glucagon receptor  Academic Article
• Covalent labeling of neurotensin receptors in rat gastric fundus plasma membranes  Academic Article
• Cross-reactive cytotoxic T cells to serologically distinct vesicular stomatitis virus.  Academic Article
• Crosstalk between the thyroid hormone and peroxisome proliferator-activated receptors in regulating peroxisome proliferator-responsive genes  Academic Article
• Cytokeratin 18 Is Expressed on the Hepatocyte Plasma Membrane Surface and Interacts with Thrombin-Antithrombin Complexes  Academic Article
• Delineation of key XRCC4/Ligase IV interfaces for targeted disruption of non-homologous end joining DNA repair  Academic Article
• Design, Synthesis, and Dopamine Receptor Modulating Activity of Spiro Bicyclic Peptidomimetics ofl-Prolyl-l-leucyl-glycinamide  Academic Article
• Determinants for calcitonin analog interaction with the calcitonin receptor N-terminus and transmembrane-loop regions.  Academic Article
• Differential acid stabilities of citraconylated amino groups of glucagon Preparation of Nα-Citraconyl glucagon and evaluation of its biological properties  Academic Article
• Differential inhibitory effects of melatonin analogs and three naphthalenic ligands on 2-[125I]iodomelatonin binding to chicken tissues  Academic Article
• Discovery of nonxanthine adenosine A2A receptor antagonists for the treatment of Parkinson's disease  Academic Article
• Dissociation of contraction and muscarinic receptor binding to isolated smooth muscle cells  Academic Article
• Distribution and characterization of vasoactive intestinal polypeptide binding in canine lower esophageal sphincter  Academic Article
• Distribution of opioid receptors in canine small intestine: implications for function  Academic Article
• Distribution of vasoactive intestinal polypeptide (VIP) binding in circular muscle and characterization of VIP binding in canine small intestinal mucosa.  Academic Article
• Divergent structural requirements exist for calcitonin receptor binding specificity and adenylate cyclase activation.  Academic Article
• Drugs???some basic concepts  Academic Article
• Dual nature of the hepatic lectin pathway for human asialotransferrin type 3 in the rat.  Academic Article
• Effect of specific trinitrophenylation of the lysine epsilon amino group of glucagon on receptor binding and adenylate cyclase activation  Academic Article
• Eliminating Competition: Characterizing and Eliminating Competitive Binding at Separate Sites between DAHP Synthase’s Essential Metal Ion and the Inhibitor DAHP Oxime  Academic Article
• Epitope specificity plays a critical role in regulating antibody-dependent cell-mediated cytotoxicity against influenza A virus  Academic Article
• Erythrocyte insulin receptors remain intact through three days of storage  Academic Article
• Evidence for Allosteric Linkage between Exosites 1 and 2 of Thrombin  Academic Article
• Evidence for Calcitonin Receptor Heterogeneity: Binding Studies with Nonhelical Analogs*  Academic Article
• Functional characterization of estrogen receptor subtypes, ERα and ERβ, mediating vitellogenin production in the liver of rainbow trout  Academic Article
• HD1, a Thrombin-directed Aptamer, Binds Exosite 1 on Prothrombin with High Affinity and Inhibits Its Activation by Prothrombinase  Academic Article
• HPLC-purified 2-[125I]iodomelatonin labels multiple binding sites in hamster brain  Academic Article
• Heterogeneity of motilin receptors in the gastrointestinal tract of the rabbit  Academic Article
• High throughput screening identifies novel inhibitors of Escherichia coli dihydrofolate reductase that are competitive with dihydrofolate  Academic Article
• High- and low-affinity states of dopamine D1 receptors in schizophrenia  Academic Article
• Histidine-rich glycoprotein binds DNA and RNA and attenuates their capacity to activate the intrinsic coagulation pathway  Academic Article
• Identification and Characterization of New Inhibitors of Fungal Homoserine Kinase  Academic Article
• Identification and characterization of high-affinity Ca2+-ATPase associated with axonal plasma membranes of dog mesenteric nerves  Academic Article
• Identification and characterization of presynaptic and postsynaptic beta adrenoreceptors in the longitudinal smooth muscle/myenteric plexus of dog ileum.  Academic Article
• Identification of Immunoglobulin Class and Subclass of House Monoclonal Antibodies to Human Cell Surface Antigens by Mixed Hemadsorption Assay  Academic Article
• Identification of novel catecholamine absorbing proteins in the central nervous system  Academic Article
• Identification of α2-adrenergic receptor sites in human retinoblastoma (Y-79) and neuroblastoma (SH-SY5Y) cells  Academic Article
• Inhibition of the amplification reactions of blood coagulation by site-specific inhibitors of α-thrombin  Academic Article
• Inhibitory effects of amiloride on alpha adrenoceptors in canine vascular smooth muscle.  Academic Article
• Insights into the unusual alpha adrenoceptor subtype in dog saphenous vein using phenoxybenzamine.  Academic Article
• Interaction of histidine-rich glycoprotein with human T lymphocytes.  Academic Article
• Investigation of α1-adrenoceptor subtypes in canine aorta, using alkylating agents  Academic Article
• Iron promotes cadmium binding to citrate.  Academic Article
• Like Fibrin, (DD)E, the Major Degradation Product of Crosslinked Fibrin, Protects Plasmin from Inhibition by α2-antiplasmin  Academic Article
• Lithium and rhythms of beta-adrenergic ([3H]CGP-12177) binding in intact rat retina, pineal gland, and hypothalamus  Academic Article
• Lowering of plasma isoxicam concentrations with acetylsalicylic acid.  Academic Article
• Lymphocyte 3H-spiroperidol binding in schizophrenia: preliminary findings  Academic Article
• MDMA-evoked changes in the binding of dopamine D2receptor ligands in striatum of rats with unilateral serotonin depletion  Academic Article
• Mannose 6-Phosphate/Insulin-like Growth Factor II Receptor Is a Death Receptor for Granzyme B during Cytotoxic T Cell–Induced Apoptosis  Academic Article
• Mapping Hsp47 binding site(s) using CNBr peptides derived from type I and type II collagen  Academic Article
• Mechanism of action of the novel plasma membrane Ca2+-pump inhibitor caloxin  Academic Article
• Melatonin Interaction with the Benzodiazepine-GABA Receptor Complex in the CNS  Academic Article
• Melatonin receptors on human granulosa cell membranes.  Academic Article
• Modulation of Agonist Binding to Human Dopamine Receptor Subtypes by l-Prolyl-l-leucyl-glycinamide and a Peptidomimetic Analog  Academic Article
• Modulation of high-affinity CNS dopamine D2 receptor by l-pro-l-leu-glycinamide (PLG) analogue  Conference Paper
• Molecular mechanism of VanHst, an alpha-ketoacid dehydrogenase required for glycopeptide antibiotic resistance from a glycopeptide producing organism  Academic Article
• Molecular requirements for inhibition of the chemokine receptor CCR8 - probe-dependent allosteric interactions  Academic Article
• Monoclonal antibodies to Escherichia coli F1-ATPase. Correlation of binding site location with interspecies cross-reactivity and effects on enzyme activity.  Academic Article
• Multimerin 1 binds factor V and activated factor V with high affinity and inhibits thrombin generation  Academic Article
• Muscarinic cholonoceptors in the rabbits myometrium: A study of the relationship between binding and response  Academic Article
• Mutagenesis and peptide analysis of the DRY motif in the α2A adrenergic receptor: evidence for alternate mechanisms in G protein-coupled receptors  Academic Article
• Neuroimaging of mirtazapine enantiomers in humans  Academic Article
• Noxious stimulation decreases substance P binding in rat spinal dorsal horn  Academic Article
• Nucleotide Selectivity of Antibiotic Kinases  Academic Article
• Occupational asthma from nickel sensitivity: I. Human serum albumin in the antigenic determinant.  Academic Article
• Occupational asthma from nickel sensitivity: II. Factors influencing the interaction of Ni2+, HSA, and serum antibodies with nickel related specificity.  Academic Article
• Oncostatin M Stimulates c-Fos to Bind a Transcriptionally Responsive AP-1 Element within the Tissue Inhibitor of Metalloproteinase-1 Promoter  Academic Article
• Opioid receptors in human neuroblastoma SH-SY5Y cells: Evidence for distinct morphine (μ) and enkephalin (δ) binding sites  Academic Article
• Overexpression, Purification, and Characterization of VanX, a D-, D-Dipeptidase which Is Essential for Vancomycin Resistance in Enterococcus faecium BM4147  Academic Article
• Peptide YY receptor in submucosal and myenteric plexus synaptosomes of canine small intestine  Academic Article
• Pharmacological characterization of melatonin binding sites in Syrian hamster hypothalamus  Academic Article
• Pharmacology of montelukast sodium (Singulair™), a potent and selective leukotriene D4 receptor antagonist  Academic Article
• Platelet-melanoma cell interaction is mediated by the glycoprotein IIb- IIIa complex  Academic Article
• Polyphosphate binds with high affinity to exosite II of thrombin  Academic Article
• Prejunctional muscarinic receptors in the deep muscular plexus of canine ileum: comparison with smooth muscle receptors.  Academic Article
• Presynaptic and postjunctional muscarinic receptors in dog ileum: binding studies  Academic Article
• Protean effects of a natural peptide agonist of the G protein-coupled secretin receptor demonstrated by receptor mutagenesis.  Academic Article
• Proton pump inhibitors: the beginning of the end or the end of the beginning?  Academic Article
• Purification of bovine striatal dopamine D-2 receptor by affinity chromatography.  Academic Article
• Quantitative autoradiography of ligands for dopamine receptors and transporters in brain of Göttingen minipig: Comparison with results in vivo  Academic Article
• Reconstitution of affinity-purified dopamine D2 receptor binding activities by specific lipids  Academic Article
• Roles of Low Specificity and Cofactor Interaction Sites on Thrombin during Factor XIII Activation  Academic Article
• Solubilization and reconstitution of dopamine D1 receptor from bovine striatal membranes: Effects of agonist and antagonist pretreatment  Academic Article
• Soluble Receptors Neutralizing TNF-α and IL-1 Block Stress-Triggered Murine Abortion  Academic Article
• Specific [3H]-guanosine binding sites in rat brain membranes  Academic Article
• Specific binding of photoaffinity-labeling peptidomimetics of Pro-Leu-Gly-NH2 to the dopamine D2L receptor: Evidence for the allosteric modulation of the dopamine receptor  Academic Article
• Specific high-affinity receptors for neurotrophin-3 on sympathetic neurons  Academic Article
• Specificity of in vitro cytotoxic T cell clones directed against vesicular stomatitis virus.  Academic Article
• Structural and Functional Interaction between the Human DNA Repair Proteins DNA Ligase IV and XRCC4  Academic Article
• Structure of the Cytoplasmic Region of PelD, a Degenerate Diguanylate Cyclase Receptor That Regulates Exopolysaccharide Production inPseudomonas aeruginosa  Academic Article
• Subtype- and response element-dependent differences in transactivation by peroxisome proliferator-activated receptors α and γ  Academic Article
• Synthesis and Structure–Activity Relationships of the First Ferrocenyl-Aryl-Hydantoin Derivatives of the Nonsteroidal Antiandrogen Nilutamide  Academic Article
• The Peroxisome Proliferator Response Element of the Gene Encoding the Peroxisomal β-Oxidation Enzyme Enoyl-CoA Hydratase/3-Hydroxyacyl-CoA Dehydrogenase Is a Target for Constitutive Androstane Receptor β/9-cis-Retinoic Acid Receptor-mediated Transactivation  Academic Article
• The direct binding of human factor VII in plasma to recombinant human tissue factor  Academic Article
• The hypersensitivity to thrombin of platelets from diabetic rats is not due to increased thrombin binding  Academic Article
• The p120ctn-binding partner Kaiso is a bi-modal DNA-binding protein that recognizes both a sequence-specific consensus and methylated CpG dinucleotides  Academic Article
• The purified myxoma virus gamma interferon receptor homolog M-T7 interacts with the heparin-binding domains of chemokines.  Academic Article
• The relationship between D 2 receptor occupancy and plasma levels on low dose oral haloperidol: a PET study  Academic Article
• UDP-N-acetylmuramic Acid (UDP-MurNAc) Is a Potent Inhibitor of MurA (Enolpyruvyl-UDP-GlcNAc Synthase)†  Academic Article
• Unusual αadrenoceptor subtype in canine saphenous vein: comparison to mesenteric vein  Academic Article
• Use of a synthetic homologue of human fibrinopeptide A for production of a monoclonal antibody specific for the free peptide.  Academic Article
• VIP receptors on canine submucosal synaptosomes  Academic Article
• Vascular effects of tetramethylpyrazuie: direct interaction with smooth muscle α-adrenoceptors  Academic Article
• Zn2+Mediates High Affinity Binding of Heparin to the αC Domain of Fibrinogen  Academic Article
• [3H] Melatonin Binding in Membrane and Cytosol Fractions From Rat and Calf Brain  Academic Article
• ets‐1 is transcriptionally up‐regulated by H 2 O 2 via an antioxidant response element  Academic Article
• α2-Adrenergic receptors on the circular smooth muscle of canine small intestine  Academic Article
• β-Amyloid efflux mediated by p-glycoprotein  Academic Article