Binding, Competitive Concept

subject area of

• 2-[¹²⁵I]Iodomelatonin Binding in the Brains of Four Salmonids  Journal Articles
• 2-[125I]Iodomelatonin binding sites in the quail heart: Characteristics, distribution and modulation by guanine nucleotides and cations  Journal Articles
• 3H-spiroperidol binding and dopamine-stimulated adenylate cyclase: Evidence for multiple classes of receptors in primate brain regions  Journal Articles
• ets‐1is transcriptionally up‐regulated by H₂O₂via an antioxidant response element  Journal Articles
• A Model for Agonism and Antagonism in an Ancient and Ubiquitous cAMP-binding Domain  Journal Articles
• A PET study of effects of chronic 3,4‐methylenedioxymethamphetamine (MDMA, “ecstasy”) on serotonin markers in Göttingen minipig brain  Journal Articles
• A molecular defect in two families with hemolytic poikilocytic anemia: reduction of high affinity membrane binding sites for ankyrin.  Journal Articles
• A simple and efficient method for solubilization of the dopamine receptor  Journal Articles
• A simple and rapid competitive enzyme‐linked immunosorbent assay to identify HPA‐1a (Pl^A1)‐negative donor platelet units  Journal Articles
• A study of phosphoglycerate kinase in human erythrocytes  Journal Articles
• Activation of protein C and thrombin activable fibrinolysis inhibitor on cultured human endothelial cells  Journal Articles
• Active suppression of host-vs graft reaction in pregnant mice. IX. Soluble suppressor activity obtained from allopregnant mouse decidua that blocks the cytolytic effector response to IL-2 is related to transforming growth factor-beta.  Journal Articles
• Active suppression of host-vs-graft reaction in pregnant mice. VI. Soluble suppressor activity obtained from decidua of allopregnant mice blocks the response to IL 2.  Journal Articles
• Agonist binding fraction of dopamine D2/3 receptors in rat brain: A quantitative autoradiographic study  Journal Articles
• Allosteric Modulation of the Dopamine D₂ Receptor by Pro-Leu-Gly-NH₂ Peptidomimetics Constrained in Either a Polyproline II Helix or a Type II β-Turn Conformation  Journal Articles
• Alpha-2 adrenoceptors on nerves and muscles of rat uterus.  Journal Articles
• Amperometric immunosensor based on polypyrrole/poly(m-pheylenediamine) multilayer on glassy carbon electrode for cytokinin N6-(Δ2-isopentenyl) adenosine assay  Journal Articles
• Analysis of Prostaglandin G/H Synthase-2 Inhibition Using Peroxidase-Induced Luminol Luminescence  Journal Articles
• Binding Sites for 2-[¹²⁵I]Iodomelatonin in the Adrenal Gland  Journal Articles
• Binding of ¹²⁵I-labelled human chorionic gonadotropin to cell membrane receptors in rabbit ovarian slices  Journal Articles
• Calcium channel antagonist binding and pharmacology in rat uterine smooth muscle  Journal Articles
• Calpain proteolysis of von Willebrand factor enhances its binding to platelet membrane glycoprotein IIb/IIIa: an explanation for platelet aggregation in thrombotic thrombocytopenic purpura  Journal Articles
• Carbohydrate-binding Modules Recognize Fine Substructures of Cellulose  Journal Articles
• Characteristics of [3H] propyl beta-carboline-3-carboxylate binding to benzodiazepine receptors in human brain.  Journal Articles
• Characterization of High‐Affinity Dopamine D₂ Receptors and Modulation of Affinity States by Guanine Nucleotides in Cholate‐Solubilized Bovine Striatal Preparations  Journal Articles
• Characterization of [3H]Ryanodine Binding Sites in Smooth Muscle of Dog Mesentery Artery  Journal Articles
• Characterization of alpha 2 adrenoceptors and other adrenoceptors in membranes isolated from dog mesenteric nerve axons.  Journal Articles
• Characterization of the prostanoid TP receptor population in human nonpregnant myometrium.  Journal Articles
• Characterization of α-Adrenoceptors in Canine Mesenteric Vein  Journal Articles
• Combination plots as graphical tools in the study of enzyme inhibition  Journal Articles
• Comparative pharmacological properties and functional coupling of mu and delta opioid receptor sites in human neuroblastoma SH-SY5Y cells.  Journal Articles
• Comparison of the Pharmacological Characteristics of 2-[¹²⁵I]Iodomelatonin Binding Sites in the Lung, Spleen, Brain and Kidney of Chicken  Journal Articles
• Competitive Effects from an Artificial Tear Solution to Protein Adsorption  Journal Articles
• Competitive solid-phase enzyme immunoassay for melatonin in human and rat serum and rat pineal gland  Journal Articles
• Complement receptor type three (CD11b/CD18) of human polymorphonuclear leukocytes recognizes fibrinogen.  Journal Articles
• Confirmatory Testing Demonstrates That False-Positive Rates in the Chlamydiazyme Assay are Influenced by Gender and Genital Specimen Type  Journal Articles
• Covalent labeling of neurotensin receptors in rat gastric fundus plasma membranes  Journal Articles
• Crosstalk between the thyroid hormone and peroxisome proliferator-activated receptors in regulating peroxisome proliferator-responsive genes  Journal Articles
• Cytokeratin 18 Is Expressed on the Hepatocyte Plasma Membrane Surface and Interacts with Thrombin-Antithrombin Complexes  Journal Articles
• Delineation of key XRCC4/Ligase IV interfaces for targeted disruption of non-homologous end joining DNA repair  Journal Articles
• Desensitization by Antidepressants of Central Norepinephrine Receptor Systems Coupled to Adenylate Cyclase^a  Journal Articles
• Design, Synthesis, and Dopamine Receptor Modulating Activity of Spiro Bicyclic Peptidomimetics ofl-Prolyl-l-leucyl-glycinamide  Journal Articles
• Different binding sites for the neuropeptide Y Y1 antagonists 1229U91 and J-104870 on human Y1 receptors  Journal Articles
• Differential inhibitory effects of melatonin analogs and three naphthalenic ligands on 2‐[¹²⁵I]iodomelatonin binding to chicken tissues  Journal Articles
• Dissociation of contraction and muscarinic receptor binding to isolated smooth muscle cells  Journal Articles
• Distribution of opioid receptors in canine small intestine: implications for function  Journal Articles
• Drugs???some basic concepts  Journal Articles
• Dual nature of the hepatic lectin pathway for human asialotransferrin type 3 in the rat.  Journal Articles
• Eliminating Competition: Characterizing and Eliminating Competitive Binding at Separate Sites between DAHP Synthase’s Essential Metal Ion and the Inhibitor DAHP Oxime  Journal Articles
• Epitope specificity plays a critical role in regulating antibody-dependent cell-mediated cytotoxicity against influenza A virus  Journal Articles
• Erythrocyte insulin receptors remain intact through three days of storage  Journal Articles
• Evidence for Allosteric Linkage between Exosites 1 and 2 of Thrombin  Journal Articles
• Functional characterization of estrogen receptor subtypes, ERα and ERβ, mediating vitellogenin production in the liver of rainbow trout  Journal Articles
• HD1, a Thrombin-directed Aptamer, Binds Exosite 1 on Prothrombin with High Affinity and Inhibits Its Activation by Prothrombinase  Journal Articles
• HPLC-purified 2-[125I]iodomelatonin labels multiple binding sites in hamster brain  Journal Articles
• High throughput screening identifies novel inhibitors of Escherichia coli dihydrofolate reductase that are competitive with dihydrofolate  Journal Articles
• High- and low-affinity states of dopamine D1 receptors in schizophrenia  Journal Articles
• Histidine-rich glycoprotein binds DNA and RNA and attenuates their capacity to activate the intrinsic coagulation pathway  Journal Articles
• Identification and Characterization of New Inhibitors of Fungal Homoserine Kinase  Journal Articles
• Identification and characterization of high-affinity Ca2+-ATPase associated with axonal plasma membranes of dog mesenteric nerves  Journal Articles
• Identification and characterization of presynaptic and postsynaptic beta adrenoreceptors in the longitudinal smooth muscle/myenteric plexus of dog ileum.  Journal Articles
• Identification of novel catecholamine absorbing proteins in the central nervous system  Journal Articles
• Identification of α2-adrenergic receptor sites in human retinoblastoma (Y-79) and neuroblastoma (SH-SY5Y) cells  Journal Articles
• Inhibition of the amplification reactions of blood coagulation by site-specific inhibitors of α-thrombin  Journal Articles
• Inhibitory effects of amiloride on alpha adrenoceptors in canine vascular smooth muscle.  Journal Articles
• Insertion of a Structural Domain of Interleukin (IL)-1β Confers Agonist Activity to the IL-1 Receptor Antagonist  Journal Articles
• Insights into the unusual alpha adrenoceptor subtype in dog saphenous vein using phenoxybenzamine.  Journal Articles
• Investigation of α₁-adrenoceptor subtypes in canine aorta, using alkylating agents  Journal Articles
• Iron promotes cadmium binding to citrate.  Journal Articles
• Like Fibrin, (DD)E, the Major Degradation Product of Crosslinked Fibrin, Protects Plasmin from Inhibition by α2-antiplasmin  Journal Articles
• Lithium and rhythms of beta-adrenergic ([3H]CGP-12177) binding in intact rat retina, pineal gland, and hypothalamus  Journal Articles
• Lowering of plasma isoxicam concentrations with acetylsalicylic acid.  Journal Articles
• Lymphocyte 3H-spiroperidol binding in schizophrenia: preliminary findings  Journal Articles
• MDMA-evoked changes in the binding of dopamine D₂receptor ligands in striatum of rats with unilateral serotonin depletion  Journal Articles
• Mannose 6-Phosphate/Insulin-like Growth Factor II Receptor Is a Death Receptor for Granzyme B during Cytotoxic T Cell–Induced Apoptosis  Journal Articles
• Mapping Hsp47 binding site(s) using CNBr peptides derived from type I and type II collagen  Journal Articles
• Mechanism of action of the novel plasma membrane Ca2+-pump inhibitor caloxin  Journal Articles
• Melatonin Interaction with the Benzodiazepine-GABA Receptor Complex in the CNS  Journal Articles
• Melatonin receptors on human granulosa cell membranes.  Journal Articles
• Method for Quantitation of Low-Abundance Nerve Growth Factor mRNA Expression in Human Nervous Tissue Using Competitive Reverse Transcription Polymerase Chain Reaction  Journal Articles
• Modulation of Agonist Binding to Human Dopamine Receptor Subtypes by l-Prolyl-l-leucyl-glycinamide and a Peptidomimetic Analog  Journal Articles
• Modulation of high-affinity CNS dopamine D2 receptor by l-pro-l-leu-glycinamide (PLG) analogue  Conferences
• Molecular mechanism of VanHst, an alpha-ketoacid dehydrogenase required for glycopeptide antibiotic resistance from a glycopeptide producing organism  Journal Articles
• Monoclonal antibodies to Escherichia coli F1-ATPase. Correlation of binding site location with interspecies cross-reactivity and effects on enzyme activity.  Journal Articles
• Multimerin 1 binds factor V and activated factor V with high affinity and inhibits thrombin generation  Journal Articles
• Muscarinic cholonoceptors in the rabbits myometrium: A study of the relationship between binding and response  Journal Articles
• Mutagenesis and peptide analysis of the DRY motif in the α2A adrenergic receptor: evidence for alternate mechanisms in G protein-coupled receptors  Journal Articles
• Neuroimaging of mirtazapine enantiomers in humans  Journal Articles
• Noxious stimulation decreases substance P binding in rat spinal dorsal horn  Journal Articles
• Nucleotide Selectivity of Antibiotic Kinases  Journal Articles
• Occupational asthma from nickel sensitivity: I. Human serum albumin in the antigenic determinant.  Journal Articles
• Occupational asthma from nickel sensitivity: II. Factors influencing the interaction of Ni2+, HSA, and serum antibodies with nickel related specificity.  Journal Articles
• Oncostatin M Stimulates c-Fos to Bind a Transcriptionally Responsive AP-1 Element within the Tissue Inhibitor of Metalloproteinase-1 Promoter  Journal Articles
• Opioid receptors in human neuroblastoma SH-SY5Y cells: Evidence for distinct morphine (μ) and enkephalin (δ) binding sites  Journal Articles
• Overexpression, Purification, and Characterization of VanX, a D-, D-Dipeptidase which Is Essential for Vancomycin Resistance in Enterococcus faecium BM4147  Journal Articles
• Pharmacological characterization of melatonin binding sites in Syrian hamster hypothalamus  Journal Articles
• Pharmacology of montelukast sodium (Singulair™), a potent and selective leukotriene D₄receptor antagonist  Journal Articles
• Prejunctional muscarinic receptors in the deep muscular plexus of canine ileum: comparison with smooth muscle receptors.  Journal Articles
• Presynaptic and postjunctional muscarinic receptors in dog ileum: binding studies  Journal Articles
• Protean effects of a natural peptide agonist of the G protein-coupled secretin receptor demonstrated by receptor mutagenesis.  Journal Articles
• Proton pump inhibitors: the beginning of the end or the end of the beginning?  Journal Articles
• Purification of bovine striatal dopamine D-2 receptor by affinity chromatography.  Journal Articles
• Quantitative autoradiography of ligands for dopamine receptors and transporters in brain of Göttingen minipig: Comparison with results in vivo  Journal Articles
• Reconstitution of affinity-purified dopamine D2 receptor binding activities by specific lipids  Journal Articles
• Selective influence of ergot alkaloids on cortical and striatal dopaminergic and sergotonergic receptors.  Journal Articles
• Solubilization and reconstitution of dopamine D1 receptor from bovine striatal membranes: Effects of agonist and antagonist pretreatment  Journal Articles
• Soluble Receptors Neutralizing TNF‐α and IL‐1 Block Stress‐Triggered Murine Abortion  Journal Articles
• Specific [³H]‐guanosine binding sites in rat brain membranes  Journal Articles
• Specific binding of photoaffinity-labeling peptidomimetics of Pro-Leu-Gly-NH2 to the dopamine D2L receptor: Evidence for the allosteric modulation of the dopamine receptor  Journal Articles
• Structural and Functional Interaction between the Human DNA Repair Proteins DNA Ligase IV and XRCC4  Journal Articles
• Structure of the Cytoplasmic Region of PelD, a Degenerate Diguanylate Cyclase Receptor That Regulates Exopolysaccharide Production in Pseudomonas aeruginosa  Journal Articles
• Subtype- and response element-dependent differences in transactivation by peroxisome proliferator-activated receptors α and γ  Journal Articles
• Synthesis and Structure–Activity Relationships of the First Ferrocenyl-Aryl-Hydantoin Derivatives of the Nonsteroidal Antiandrogen Nilutamide  Journal Articles
• Systematic replacement of amides by 1,4-disubstituted[1,2,3]triazoles in Leu-enkephalin and the impact on the delta opioid receptor activity.  Journal Articles
• The Peroxisome Proliferator Response Element of the Gene Encoding the Peroxisomal β-Oxidation Enzyme Enoyl-CoA Hydratase/3-Hydroxyacyl-CoA Dehydrogenase Is a Target for Constitutive Androstane Receptor β/9-cis-Retinoic Acid Receptor-mediated Transactivation  Journal Articles
• The direct binding of human factor VII in plasma to recombinant human tissue factor  Journal Articles
• The hypersensitivity to thrombin of platelets from diabetic rats is not due to increased thrombin binding  Journal Articles
• The p120ctn-binding partner Kaiso is a bi-modal DNA-binding protein that recognizes both a sequence-specific consensus and methylated CpG dinucleotides  Journal Articles
• The purified myxoma virus gamma interferon receptor homolog M-T7 interacts with the heparin-binding domains of chemokines  Journal Articles
• UDP-N-acetylmuramic Acid (UDP-MurNAc) Is a Potent Inhibitor of MurA (Enolpyruvyl-UDP-GlcNAc Synthase)  Journal Articles
• Unusual αadrenoceptor subtype in canine saphenous vein: comparison to mesenteric vein  Journal Articles
• Use of a synthetic homologue of human fibrinopeptide A for production of a monoclonal antibody specific for the free peptide  Journal Articles
• Vascular effects of tetramethylpyrazuie: direct interaction with smooth muscle α-adrenoceptors  Journal Articles
• Zn2+ Mediates High Affinity Binding of Heparin to the αC Domain of Fibrinogen  Journal Articles
• [³H] Melatonin Binding in Membrane and Cytosol Fractions From Rat and Calf Brain  Journal Articles