Binding, Competitive
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Overview
subject area of
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2-(Oxadiazolyl)- and 2-(thiazolyl)imidazo[1,2-a]pyrimidines as agonists and inverse agonists at benzodiazepine receptors Academic Article
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2-[125I]Iodomelatonin binding sites in the quail heart: Characteristics, distribution and modulation by guanine nucleotides and cations Academic Article
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2-[125I]Iodomelatonin Binding in the Brains of Four Salmonids Academic Article
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3H-spiroperidol binding and dopamine-stimulated adenylate cyclase: Evidence for multiple classes of receptors in primate brain regions Academic Article
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A Model for Agonism and Antagonism in an Ancient and Ubiquitous cAMP-binding Domain Academic Article
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A PET study of effects of chronic 3,4-methylenedioxymethamphetamine (MDMA, “ecstasy”) on serotonin markers in Göttingen minipig brain Academic Article
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A molecular defect in two families with hemolytic poikilocytic anemia: reduction of high affinity membrane binding sites for ankyrin. Academic Article
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A simple and efficient method for solubilization of the dopamine receptor Academic Article
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A simple and rapid competitive enzyme-linked immunosorbent assay to identify HPA-1a (PlA1)-negative donor platelet units Academic Article
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A study of phosphoglycerate kinase in human erythrocytes Academic Article
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Activation of a recombinant human factor VII structural analogue alters its affinity of binding to tissue factor Academic Article
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Activation of protein C and thrombin activable fibrinolysis inhibitor on cultured human endothelial cells Academic Article
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Active suppression of host-vs graft reaction in pregnant mice. IX. Soluble suppressor activity obtained from allopregnant mouse decidua that blocks the cytolytic effector response to IL-2 is related to transforming growth factor-beta. Academic Article
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Active suppression of host-vs-graft reaction in pregnant mice. VI. Soluble suppressor activity obtained from decidua of allopregnant mice blocks the response to IL 2. Academic Article
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Agonist binding fraction of dopamine D2/3 receptors in rat brain: A quantitative autoradiographic study Academic Article
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Agonists Interaction with Radiolabeled α-Adrenoceptor Antagonists Binding Sites in Rat Mesenteric Artery Academic Article
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Allosteric Modulation of the Dopamine D2Receptor by Pro-Leu-Gly-NH2Peptidomimetics Constrained in Either a Polyproline II Helix or a Type II β-Turn Conformation Academic Article
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Alpha-2 adrenoceptors on nerves and muscles of rat uterus. Academic Article
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Binding Sites for 2-[125I]Iodomelatonin in the Adrenal Gland Academic Article
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Binding of 125I-labelled human chorionic gonadotropin to cell membrane receptors in rabbit ovarian slices Academic Article
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Biochemical studies on opioid and alpha 2-adrenergic receptors in canine submucosal neurons Academic Article
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Calcium channel antagonist binding and pharmacology in rat uterine smooth muscle Academic Article
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Calpain proteolysis of von Willebrand factor enhances its binding to platelet membrane glycoprotein IIb/IIIa: an explanation for platelet aggregation in thrombotic thrombocytopenic purpura Academic Article
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Carbohydrate-binding Modules Recognize Fine Substructures of Cellulose Academic Article
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Characteristics of [3H] propyl beta-carboline-3-carboxylate binding to benzodiazepine receptors in human brain. Academic Article
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Characterization of High-Affinity Dopamine D2Receptors and Modulation of Affinity States by Guanine Nucleotides in Cholate-Solubilized Bovine Striatal Preparations Academic Article
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Characterization of [3H]Ryanodine Binding Sites in Smooth Muscle of Dog Mesentery Artery Academic Article
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Characterization of alpha 2 adrenoceptors and other adrenoceptors in membranes isolated from dog mesenteric nerve axons. Academic Article
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Characterization of beta adrenoceptors on cultured endothelial cells by radioligand binding Academic Article
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Characterization of cholecystokinin receptors in canine intestinal circular muscle Academic Article
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Characterization of galanin receptor in canine small intestinal circular muscle synaptosomes Academic Article
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Characterization of neurokinin type 1 receptor in canine small intestinal muscle Academic Article
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Characterization of the prostanoid TP receptor population in human nonpregnant myometrium. Academic Article
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Characterization of α-Adrenoceptors in Canine Mesenteric Vein Academic Article
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Combination plots as graphical tools in the study of enzyme inhibition Academic Article
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Comparative pharmacological properties and functional coupling of mu and delta opioid receptor sites in human neuroblastoma SH-SY5Y cells. Academic Article
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Comparison of the Pharmacological Characteristics of 2-[125I]Iodomelatonin Binding Sites in the Lung, Spleen, Brain and Kidney of Chicken Academic Article
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Competitive Effects from an Artificial Tear Solution to Protein Adsorption Academic Article
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Competitive solid-phase enzyme immunoassay for melatonin in human and rat serum and rat pineal gland. Academic Article
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Complement receptor type three (CD11b/CD18) of human polymorphonuclear leukocytes recognizes fibrinogen. Academic Article
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Complex formation of platelet thrombospondin with fibrinogen. Academic Article
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Complex formation of platelet thrombospondin with histidine-rich glycoprotein. Academic Article
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Confirmatory Testing Demonstrates That False-Positive Rates in the Chlamydiazyme Assay are Influenced by Gender and Genital Specimen Type Academic Article
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Conformational determinants in receptor recognition of peptide hormones: interaction of parathyroid hormone with the glucagon receptor Academic Article
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Covalent labeling of neurotensin receptors in rat gastric fundus plasma membranes Academic Article
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Crosstalk between the thyroid hormone and peroxisome proliferator-activated receptors in regulating peroxisome proliferator-responsive genes Academic Article
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Cytokeratin 18 Is Expressed on the Hepatocyte Plasma Membrane Surface and Interacts with Thrombin-Antithrombin Complexes Academic Article
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Delineation of key XRCC4/Ligase IV interfaces for targeted disruption of non-homologous end joining DNA repair Academic Article
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Design, Synthesis, and Dopamine Receptor Modulating Activity of Spiro Bicyclic Peptidomimetics ofl-Prolyl-l-leucyl-glycinamide Academic Article
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Determinants for calcitonin analog interaction with the calcitonin receptor N-terminus and transmembrane-loop regions. Academic Article
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Differential acid stabilities of citraconylated amino groups of glucagon Preparation of Nα-Citraconyl glucagon and evaluation of its biological properties Academic Article
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Differential inhibitory effects of melatonin analogs and three naphthalenic ligands on 2-[125I]iodomelatonin binding to chicken tissues Academic Article
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Discovery of nonxanthine adenosine A2A receptor antagonists for the treatment of Parkinson's disease Academic Article
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Dissociation of contraction and muscarinic receptor binding to isolated smooth muscle cells Academic Article
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Distribution and characterization of vasoactive intestinal polypeptide binding in canine lower esophageal sphincter Academic Article
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Distribution of opioid receptors in canine small intestine: implications for function Academic Article
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Distribution of vasoactive intestinal polypeptide (VIP) binding in circular muscle and characterization of VIP binding in canine small intestinal mucosa. Academic Article
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Divergent structural requirements exist for calcitonin receptor binding specificity and adenylate cyclase activation. Academic Article
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Drugs???some basic concepts Academic Article
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Dual nature of the hepatic lectin pathway for human asialotransferrin type 3 in the rat. Academic Article
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Effect of specific trinitrophenylation of the lysine epsilon amino group of glucagon on receptor binding and adenylate cyclase activation Academic Article
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Eliminating Competition: Characterizing and Eliminating Competitive Binding at Separate Sites between DAHP Synthase’s Essential Metal Ion and the Inhibitor DAHP Oxime Academic Article
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Epitope specificity plays a critical role in regulating antibody-dependent cell-mediated cytotoxicity against influenza A virus Academic Article
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Erythrocyte insulin receptors remain intact through three days of storage Academic Article
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Evidence for Allosteric Linkage between Exosites 1 and 2 of Thrombin Academic Article
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Evidence for Calcitonin Receptor Heterogeneity: Binding Studies with Nonhelical Analogs* Academic Article
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Functional characterization of estrogen receptor subtypes, ERα and ERβ, mediating vitellogenin production in the liver of rainbow trout Academic Article
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HD1, a Thrombin-directed Aptamer, Binds Exosite 1 on Prothrombin with High Affinity and Inhibits Its Activation by Prothrombinase Academic Article
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HPLC-purified 2-[125I]iodomelatonin labels multiple binding sites in hamster brain Academic Article
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Heterogeneity of motilin receptors in the gastrointestinal tract of the rabbit Academic Article
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High throughput screening identifies novel inhibitors of Escherichia coli dihydrofolate reductase that are competitive with dihydrofolate Academic Article
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High- and low-affinity states of dopamine D1 receptors in schizophrenia Academic Article
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Histidine-rich glycoprotein binds DNA and RNA and attenuates their capacity to activate the intrinsic coagulation pathway Academic Article
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Identification and Characterization of New Inhibitors of Fungal Homoserine Kinase Academic Article
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Identification and characterization of high-affinity Ca2+-ATPase associated with axonal plasma membranes of dog mesenteric nerves Academic Article
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Identification and characterization of presynaptic and postsynaptic beta adrenoreceptors in the longitudinal smooth muscle/myenteric plexus of dog ileum. Academic Article
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Identification of Immunoglobulin Class and Subclass of House Monoclonal Antibodies to Human Cell Surface Antigens by Mixed Hemadsorption Assay Academic Article
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Identification of novel catecholamine absorbing proteins in the central nervous system Academic Article
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Identification of α2-adrenergic receptor sites in human retinoblastoma (Y-79) and neuroblastoma (SH-SY5Y) cells Academic Article
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Inhibition of the amplification reactions of blood coagulation by site-specific inhibitors of α-thrombin Academic Article
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Inhibitory effects of amiloride on alpha adrenoceptors in canine vascular smooth muscle. Academic Article
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Insights into the unusual alpha adrenoceptor subtype in dog saphenous vein using phenoxybenzamine. Academic Article
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Interaction of histidine-rich glycoprotein with human T lymphocytes. Academic Article
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Investigation of α1-adrenoceptor subtypes in canine aorta, using alkylating agents Academic Article
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Iron promotes cadmium binding to citrate. Academic Article
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Like Fibrin, (DD)E, the Major Degradation Product of Crosslinked Fibrin, Protects Plasmin from Inhibition by α2-antiplasmin Academic Article
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Lithium and rhythms of beta-adrenergic ([3H]CGP-12177) binding in intact rat retina, pineal gland, and hypothalamus Academic Article
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Lowering of plasma isoxicam concentrations with acetylsalicylic acid. Academic Article
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Lymphocyte 3H-spiroperidol binding in schizophrenia: preliminary findings Academic Article
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MDMA-evoked changes in the binding of dopamine D2receptor ligands in striatum of rats with unilateral serotonin depletion Academic Article
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Mannose 6-Phosphate/Insulin-like Growth Factor II Receptor Is a Death Receptor for Granzyme B during Cytotoxic T Cell–Induced Apoptosis Academic Article
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Mapping Hsp47 binding site(s) using CNBr peptides derived from type I and type II collagen Academic Article
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Mechanism of action of the novel plasma membrane Ca2+-pump inhibitor caloxin Academic Article
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Melatonin Interaction with the Benzodiazepine-GABA Receptor Complex in the CNS Academic Article
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Melatonin receptors on human granulosa cell membranes. Academic Article
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Modulation of Agonist Binding to Human Dopamine Receptor Subtypes by l-Prolyl-l-leucyl-glycinamide and a Peptidomimetic Analog Academic Article
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Modulation of high-affinity CNS dopamine D2 receptor by l-pro-l-leu-glycinamide (PLG) analogue Conference Paper
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Molecular mechanism of VanHst, an alpha-ketoacid dehydrogenase required for glycopeptide antibiotic resistance from a glycopeptide producing organism Academic Article
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Monoclonal antibodies to Escherichia coli F1-ATPase. Correlation of binding site location with interspecies cross-reactivity and effects on enzyme activity. Academic Article
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Multimerin 1 binds factor V and activated factor V with high affinity and inhibits thrombin generation Academic Article
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Muscarinic cholonoceptors in the rabbits myometrium: A study of the relationship between binding and response Academic Article
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Mutagenesis and peptide analysis of the DRY motif in the α2A adrenergic receptor: evidence for alternate mechanisms in G protein-coupled receptors Academic Article
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Neuroimaging of mirtazapine enantiomers in humans Academic Article
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Noxious stimulation decreases substance P binding in rat spinal dorsal horn Academic Article
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Nucleotide Selectivity of Antibiotic Kinases Academic Article
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Occupational asthma from nickel sensitivity: I. Human serum albumin in the antigenic determinant. Academic Article
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Occupational asthma from nickel sensitivity: II. Factors influencing the interaction of Ni2+, HSA, and serum antibodies with nickel related specificity. Academic Article
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Oncostatin M Stimulates c-Fos to Bind a Transcriptionally Responsive AP-1 Element within the Tissue Inhibitor of Metalloproteinase-1 Promoter Academic Article
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Opioid receptors in human neuroblastoma SH-SY5Y cells: Evidence for distinct morphine (μ) and enkephalin (δ) binding sites Academic Article
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Overexpression, Purification, and Characterization of VanX, a D-, D-Dipeptidase which Is Essential for Vancomycin Resistance in Enterococcus faecium BM4147 Academic Article
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Peptide YY receptor in submucosal and myenteric plexus synaptosomes of canine small intestine Academic Article
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Pharmacological characterization of melatonin binding sites in Syrian hamster hypothalamus Academic Article
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Pharmacology of montelukast sodium (Singulair™), a potent and selective leukotriene D4 receptor antagonist Academic Article
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Platelet-melanoma cell interaction is mediated by the glycoprotein IIb- IIIa complex Academic Article
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Polyphosphate binds with high affinity to exosite II of thrombin Academic Article
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Prejunctional muscarinic receptors in the deep muscular plexus of canine ileum: comparison with smooth muscle receptors. Academic Article
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Presynaptic and postjunctional muscarinic receptors in dog ileum: binding studies Academic Article
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Protean effects of a natural peptide agonist of the G protein-coupled secretin receptor demonstrated by receptor mutagenesis. Academic Article
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Proton pump inhibitors: the beginning of the end or the end of the beginning? Academic Article
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Purification of bovine striatal dopamine D-2 receptor by affinity chromatography. Academic Article
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Quantitative autoradiography of ligands for dopamine receptors and transporters in brain of Göttingen minipig: Comparison with results in vivo Academic Article
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Reconstitution of affinity-purified dopamine D2 receptor binding activities by specific lipids Academic Article
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Roles of Low Specificity and Cofactor Interaction Sites on Thrombin during Factor XIII Activation Academic Article
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Solubilization and reconstitution of dopamine D1 receptor from bovine striatal membranes: Effects of agonist and antagonist pretreatment Academic Article
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Soluble Receptors Neutralizing TNF-α and IL-1 Block Stress-Triggered Murine Abortion Academic Article
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Specific [3
H]-guanosine binding sites in rat brain membranes Academic Article
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Specific binding of photoaffinity-labeling peptidomimetics of Pro-Leu-Gly-NH2 to the dopamine D2L receptor: Evidence for the allosteric modulation of the dopamine receptor Academic Article
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Structural and Functional Interaction between the Human DNA Repair Proteins DNA Ligase IV and XRCC4 Academic Article
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Structure of the Cytoplasmic Region of PelD, a Degenerate Diguanylate Cyclase Receptor That Regulates Exopolysaccharide Production in Pseudomonas aeruginosa Academic Article
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Subtype- and response element-dependent differences in transactivation by peroxisome proliferator-activated receptors α and γ Academic Article
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Synthesis and Structure–Activity Relationships of the First Ferrocenyl-Aryl-Hydantoin Derivatives of the Nonsteroidal Antiandrogen Nilutamide Academic Article
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The Peroxisome Proliferator Response Element of the Gene Encoding the Peroxisomal β-Oxidation Enzyme Enoyl-CoA Hydratase/3-Hydroxyacyl-CoA Dehydrogenase Is a Target for Constitutive Androstane Receptor β/9-cis-Retinoic Acid Receptor-mediated Transactivation Academic Article
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The direct binding of human factor VII in plasma to recombinant human tissue factor Academic Article
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The hypersensitivity to thrombin of platelets from diabetic rats is not due to increased thrombin binding Academic Article
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The p120ctn-binding partner Kaiso is a bi-modal DNA-binding protein that recognizes both a sequence-specific consensus and methylated CpG dinucleotides Academic Article
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The purified myxoma virus gamma interferon receptor homolog M-T7 interacts with the heparin-binding domains of chemokines. Academic Article
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The relationship between D 2 receptor occupancy and plasma levels on low dose oral haloperidol: a PET study Academic Article
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UDP-N-acetylmuramic Acid (UDP-MurNAc) Is a Potent Inhibitor of MurA (Enolpyruvyl-UDP-GlcNAc Synthase)† Academic Article
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Unusual αadrenoceptor subtype in canine saphenous vein: comparison to mesenteric vein Academic Article
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Use of a synthetic homologue of human fibrinopeptide A for production of a monoclonal antibody specific for the free peptide. Academic Article
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VIP receptors on canine submucosal synaptosomes Academic Article
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Vascular effects of tetramethylpyrazuie: direct interaction with smooth muscle α-adrenoceptors Academic Article
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Zn2+ Mediates High Affinity Binding of Heparin to the αC Domain of Fibrinogen Academic Article
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[3H] Melatonin Binding in Membrane and Cytosol Fractions From Rat and Calf Brain Academic Article
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ets‐1
is transcriptionally up‐regulated by H
2
O
2
via an antioxidant response element Academic Article
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α2-Adrenergic receptors on the circular smooth muscle of canine small intestine Academic Article
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β-Amyloid efflux mediated by p-glycoprotein Academic Article