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A Phase I study of cyclin-dependent kinase...
Journal article

A Phase I study of cyclin-dependent kinase inhibitor, AT7519, in patients with advanced cancer: NCIC Clinical Trials Group IND 177

Abstract

Background:AT7519 is a small-molecular inhibitor of multiple cyclin-dependent kinases (CDKs). It shows encouraging anti-cancer activity against multiple cell lines and in tumour xenografts. This phase I study was conducted to evaluate the safety and tolerability of AT7519 given as 1-h intravenous infusion on days 1, 4, 8 and 11 every 3 weeks.Methods:Patients with advanced refractory solid tumours or non-Hodgkin’s lymphoma were enroled. Dose …

Authors

Chen EX; Hotte S; Hirte H; Siu LL; Lyons J; Squires M; Lovell S; Turner S; McIntosh L; Seymour L

Journal

British Journal of Cancer, Vol. 111, No. 12, pp. 2262–2267

Publisher

Springer Nature

Publication Date

December 2014

DOI

10.1038/bjc.2014.565

ISSN

0007-0920