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d-Ala-d-Ala carboxypeptidase VanY
Chapter

d-Ala-d-Ala carboxypeptidase VanY

Abstract

The subject of this chapter is d-ala-d-ala Carboxypeptidase VanY. The VanY carboxypeptidase releases the C-terminal hydrolyses the d-ala from the precursor peptides that provide the crosslinks in the bacterial cell wall peptidoglycans. The enzyme has been characterized from a strain of the pathogenic bacterium Enterococcus faecium that is insensitive to the antibiotic vancomycin. Vancomycin binds to the d-Ala-d-Ala portion of the crosslinking peptide, preventing a transpeptidase from making the crosslinks in the peptidoglycan. The vancomycin resistance genes are encoded on a plasmid, and the VanH and VanA proteins produce the depsipeptide d-ala-d-lactate instead of d-ala-d-Ala. VanX degrades d-ala-d-Ala, pushing the equilibrium toward d-ala-d-lactate. d-ala-d-lactate can be used to crosslink the peptidoglycan but has a lower affinity for vancomycin, hence the resistance to the antibiotic. Unlike VanX, VanY is a penicillin-binding protein and forms a stable complex with benzylpenicillin. VanY increases tolerance to vancomycin but is dispensable in the presence of the vanHAX genes.

Authors

Thaker M; Wright G

Book title

Handbook of Proteolytic Enzymes Metallopeptidases

Pagination

pp. 1659-1661

Publication Date

January 1, 2025

DOI

10.1016/B978-0-443-28849-4.00259-9
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