selected scholarly activity
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chapters
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conferences
- DEVELOPMENT OF NOVEL ANTI-BRAIN METASTASIS INHIBITORS. Neuro-Oncology. 98-99. 2022
- New alpha-thioalkyl phosphonium salts as Wittig substrates for vinyl sulfide synthesis. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2019
- Synthesis of Cannabigerol derivatives via direct ortho-allylation of phenols. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2019
- Vinyl sulfides: New preparations and reactions. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2019
- A macrophage-based screen identifies antibacterial compounds selective for intracellular Salmonella Typhimurium. 383828. 2018
- Introducing Fe-Non: A synthetic iron-rich nontronite clay for green oxidations. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2016
- Use of alumina for Luche-selective reduction of ketones. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2016
- Cerium-free Luche reduction in the presence of alumina. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2015
- Gram scale total synthesis of veranamine. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2015
- New applications of dimethylsulfoxide as a terminal oxidant. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2015
- Progress toward the total synthesis of tetarimycin A. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2015
- Synthetic clays as new catalysts for aerobic oxidation. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2015
- Efficient SNAr and nitrile hydrolysis on the surface of KF/Alumina. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2012
- Heterogeneous catalysis for procedurally efficient heterocyclic synthesis. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2012
- New applications of metal oxides for dehydrogenation chemistry. ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY. 2012
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journal articles
- Perturbation of Pseudomonas aeruginosa peptidoglycan recycling by anti-folates and design of a dual-action inhibitor.. mBio. 16:e0298424. 2025
- High-Throughput Discovery of Synthetic Siderophores for Trojan Horse Antibiotics.. ACS Infectious Diseases. 10:3821-3841. 2024
- A screen for cell envelope stress uncovers an inhibitor of prolipoprotein diacylglyceryl transferase, Lgt, in Escherichia coli.. iScience. 27:110894. 2024
- De novo GTP synthesis is a metabolic vulnerability for the interception of brain metastases.. Cell Reports Medicine. 5:101755. 2024
- TRSC-04 DE NOVO GTP SYNTHESIS IS A METABOLIC VULNERABILITY FOR THE INTERCEPTION OF BRAIN METASTASES. NOA. 6:i40-i40. 2024
- NOVEL CAFFEINE DERIVATIVES MITIGATE HYPERLIPIDEMIA BY REDUCING PCSK9 EXPRESSION AND SECRETION. Atherosclerosis. 395. 2024
- A platform for predicting mechanism of action based on bacterial transcriptional responses identifies an unusual DNA gyrase inhibitor. Cell Reports. 43:114053-114053. 2024
- Allosteric inhibition of tRNA synthetase Gln4 by N-pyrimidinyl-β-thiophenylacrylamides exerts highly selective antifungal activity. Cell Chemical Biology. 31:760-775.e17. 2024
- Deep learning-guided discovery of an antibiotic targeting Acinetobacter baumannii. Nature Chemical Biology. 19:1342-1350. 2023
- INTERCEPTING BRAIN METASTASES THROUGH METABOLIC VULNERABILITIES. NOA. 5:i2-i2. 2023
- An effective kinase inhibition strategy for metastatic recurrent childhood medulloblastoma. Journal of Neuro-Oncology. 163:635-645. 2023
- Bioactivity of the cannabigerol cannabinoid and its analogues – the role of 3-dimensional conformation. Organic and Biomolecular Chemistry. 21:4683-4693. 2023
- Abstract 2474: Uncovering a new therapeutic vulnerability for preventing brain metastases. Cancer Research. 83:2474-2474. 2023
- <i>Garcinia buchananii</i> stem bark extract and its bioactive constituents manniflavanone, GB-2 and buchananiflavanone attenuate intestinal inhibitory neuromuscular transmission. Journal of Smooth Muscle Research. 59:34-57. 2023
- DDDR-03. DEVELOPMENT OF NOVEL ANTI-BRAIN METASTASIS INHIBITORS. Neuro-Oncology. 24:vii98-vii99. 2022
- Use of Vinyl Sulfides in Fischer Indole Reactions. Synthesis. 54:4917-4931. 2022
- Genetic and Chemical Screening Reveals Targets and Compounds to Potentiate Gram-Positive Antibiotics against Gram-Negative Bacteria. ACS Infectious Diseases. 8:2187-2197. 2022
- QSAR models reveal new EPAC-selective allosteric modulators. RSC Chemical Biology. 3:1230-1239. 2022
- BSCI-13 DEVELOPMENT OF NOVEL ANTI-BRAIN METASTASIS INHIBITORS. NOA. 4:i3-i3. 2022
- Antibacterial Activity of Metergoline Analogues: Revisiting the Ergot Alkaloid Scaffold for Antibiotic Discovery. ACS Medicinal Chemistry Letters. 13:284-291. 2022
- Caffeine blocks SREBP2-induced hepatic PCSK9 expression to enhance LDLR-mediated cholesterol clearance. Nature Communications. 13:770. 2022
- Bibenzyl synthesis in Cannabis sativa L.. The Plant Journal. 109:693-707. 2022
- Exploration of BAY 11-7082 as a Potential Antibiotic. ACS Infectious Diseases. 8:170-182. 2022
- Targeting SUMOylation dependency in human cancer stem cells through a unique SAE2 motif revealed by chemical genomics. Cell Chemical Biology. 28:1394-1406.e10. 2021
- Exploration of BAY 11-7082 as a novel antibiotic 2021
- Aldehyde to Ketone Homologation Enabled by Improved Access to Thioalkyl Phosphonium Salts. Organic Letters. 23:4548-4552. 2021
- Chemical Screen for Vancomycin Antagonism Uncovers Probes of the Gram-Negative Outer Membrane. ACS Chemical Biology. 16:929-942. 2021
- Hexafluoroisopropyl Sulfamate: A Useful Reagent for the Synthesis of Sulfamates and Sulfamides. Organic Letters. 23:3373-3378. 2021
- Efficient Synthesis of Cannabigerol, Grifolin, and Piperogalin via Alumina-Promoted Allylation. Journal of natural products. 83:2587-2591. 2020
- Genetic and Chemical Screening in Human Blood Serum Reveals Unique Antibacterial Targets and Compounds against Klebsiella pneumoniae. Cell Reports. 32:107927-107927. 2020
- Targeting Two-Component Systems Uncovers a Small-Molecule Inhibitor of Salmonella Virulence. Cell Chemical Biology. 27:793-805.e7. 2020
- Mechanism of Action of an EPAC1-Selective Competitive Partial Agonist. Journal of Medicinal Chemistry. 63:4762-4775. 2020
- Isolation and Synthesis of Veranamine, an Antidepressant Lead from the Marine Sponge Verongula rigida. Journal of natural products. 83:1092-1098. 2020
- Uncovering the Hidden Antibiotic Potential of Cannabis. ACS Infectious Diseases. 6:338-346. 2020
- Alkylation of Indoles with α,β‐Unsaturated Ketones using Alumina in Hexanes. Advanced Synthesis and Catalysis. 361:5548-5551. 2019
- Uncovering the hidden antibiotic potential of Cannabis 2019
- One-pot carbonyl reduction and carbonate formation using sodium borohydride in dialkyl carbonate solvents. Tetrahedron Letters. 60:151203-151203. 2019
- A macrophage-based screen identifies antibacterial compounds selective for intracellular Salmonella Typhimurium. Nature Communications. 10:197. 2019
- ChemInform Abstract: Biaryl Ketones by Suzuki—Miyaura Cross‐Coupling of Organotrifluoroborates and Acyl Chlorides.. ChemInform. 47:no-no. 2016
- ChemInform Abstract: Cerium‐Free Luche Reduction Directed by Rehydrated Alumina.. ChemInform. 47:no-no. 2016
- Biaryl Ketones by Suzuki–Miyaura Cross‐Coupling of Organotrifluoroborates and Acyl Chlorides. European Journal of Organic Chemistry. 2016:2983-2987. 2016
- Cerium-free Luche reduction directed by rehydrated alumina. Tetrahedron. 72:3748-3753. 2016
- ChemInform Abstract: Dimethyl Sulfoxide as a Synthon in Organic Chemistry. ChemInform. 47:no-no. 2016
- Dimethyl Sulfoxide as a Synthon in Organic Chemistry. Synthesis. 48:1421-1436. 2016
- Evaluation of synthetic coumarins for antiausterity cytotoxicity against pancreatic cancers. Bioorganic and Medicinal Chemistry Letters. 26:1471-1474. 2016
- ChemInform Abstract: Bromination of Olefins with HBr and DMSO.. ChemInform. 46:no-no. 2015
- Bromination of Olefins with HBr and DMSO. Journal of Organic Chemistry. 80:3701-3707. 2015
- ChemInform Abstract: Aryl Methyl Sulfides via SNAr Using DMSO as the Source of the Thiomethyl Moiety.. ChemInform. 46:no-no. 2015
- Aryl methyl sulfides via SNAr using DMSO as the source of the thiomethyl moiety. Tetrahedron Letters. 55:5323-5326. 2014
- ChemInform Abstract: Dehydroaromatization with V2O5.. ChemInform. 44:no-no. 2013
- Dehydroaromatization with V2O5. Synlett. 24:1675-1678. 2013
- ChemInform Abstract: Combined Pd/C and Montmorillonite Catalysis for One‐Pot Synthesis of Benzimidazoles.. ChemInform. 44:no-no. 2013
- Combined Pd/C and Montmorillonite Catalysis for One‐Pot Synthesis of Benzimidazoles. European Journal of Organic Chemistry. 2012:6508-6512. 2012
- ChemInform Abstract: Directed Remote Aromatic Metalations: Mechanisms and Driving Forces. ChemInform. 43:no-no. 2012
- Synthesis and Evaluation of Anticancer Natural Product Analogues Based on Angelmarin: Targeting the Tolerance towards Nutrient Deprivation. ChemMedChem. 7:766-770. 2012
- Directed Remote Aromatic Metalations: Mechanisms and Driving Forces. Chemistry - A European Journal. 18:3804-3820. 2012
- Targeting the Resistance of Pancreatic Cancer Cells to Nutrient Deprivation: Anti-Austerity Compounds. Current Drug Delivery. 7:355-369. 2010
- ChemInform Abstract: Total Synthesis of (+)‐Angelmarin.. ChemInform. 40:no-no. 2009
- Total Synthesis of (+)-Angelmarin. Journal of Organic Chemistry. 74:5083-5086. 2009
- ChemInform Abstract: Total Synthesis of (.+‐.)‐Mersicarpine.. ChemInform. 39:no-no. 2008
- Total Synthesis of (±)-Mersicarpine. Organic Letters. 10:1437-1440. 2008
- Expanding the Scope of Mn(OAc)3‐Mediated Cyclizations: Synthesis of the Tetracyclic Core of Tronocarpine.. ChemInform. 38:no-no. 2007
- Siloxane-terminated phenylpyrimidine liquid crystal hosts. Journal of Materials Chemistry. 17:2313-2313. 2007
- Expanding the Scope of Mn(OAc)3-Mediated Cyclizations: Synthesis of the Tetracyclic Core of Tronocarpine. Organic Letters. 8:4561-4564. 2006
- Synthesis of the Western Half of the Lolicines and Lolitrems. Organic Letters. 8:2209-2212. 2006
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preprints